SCHEMBL9727409

SCHEMBL9727409

CC(C)Oc1ccc(S(=O)(=O)N2CCCC2=O)cc1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TP53 P04637 6/20 0.48
DHCR7 Q9UBM7 1/20 0.47
MMP2 P08253 2/20 0.47
GAA P10253 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
WDR5 P61964 1/20 0.42
MMP3 P08254 1/20 0.42
MMP9 P14780 1/20 0.42
MMP14 P50281 1/20 0.42
HTT P42858 2/20 0.41
POLB P06746 1/20 0.41
ALDH1A1 P00352 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042185 0.79 MMP2 (0.65) TP53MMP2MEN1KMT2AHTT
SCHEMBL7383735 0.79 MMP2 (0.64) TP53MMP2GAAMEN1KMT2A
SCHEMBL9727635 0.78 GAA (0.46) TP53MMP2GAAMEN1KMT2A
SCHEMBL12209246 0.77 HTT (0.66) DHCR7GAAMEN1KMT2AHTT
SCHEMBL9727557 0.77 GAA (0.44) TP53MMP2GAA
SCHEMBL9621784 0.77 TSHR (0.61) TP53MMP2GAAHTTALDH1A1
SCHEMBL19348522 0.77 DHCR7 (0.59) DHCR7KMT2AHTTPTGDR2
SCHEMBL16788114 0.76 HTT (0.69) DHCR7GAAMEN1KMT2AHTT
SCHEMBL7379601 0.75 MMP2 (0.64) TP53MMP2GAAMEN1KMT2A
SCHEMBL10702282 0.75 MMP2 (0.64) TP53MMP2GAAKMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5164514-A Antispasmodics ROUSSEL UCLAF (FR) 1992-11-17 US disclosed
US-5081130-A Antispasmodic agents ROUSSEL UCLAF (FR) 1992-01-14 US disclosed
US-4990531-A Antispasmodic agents ROUSSEL UCLAF (FR) 1991-02-05 US disclosed
EP-0335758-A2 Derivatives of 1-arylsulfonyl-2-pyrolidinone, process for their preparation, their use as medicaments and compositions containing them ROUSSEL-UCLAF (FR) 1989-10-04 EP disclosed