SCHEMBL9727557

SCHEMBL9727557

CC(C)Sc1ccc(S(=O)(=O)N2CCCC2=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.44
TP53 P04637 5/20 0.42
TSHR P16473 1/20 0.41
AKR1C3 P42330 4/20 0.40
MMP2 P08253 1/20 0.40
PTGDR Q13258 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727536 0.84 TSHR (0.59) GAATP53TSHRAKR1C3MMP2
SCHEMBL7383735 0.79 MMP2 (0.64) GAATP53MMP2
SCHEMBL9727635 0.78 GAA (0.46) GAATP53AKR1C3MMP2
SCHEMBL9727409 0.77 TP53 (0.48) GAATP53MMP2
SCHEMBL7379601 0.75 MMP2 (0.64) GAATP53AKR1C3MMP2
SCHEMBL10702282 0.75 MMP2 (0.64) GAATP53AKR1C3MMP2
SCHEMBL7380549 0.75 PKM (0.62) GAATP53AKR1C3MMP2
SCHEMBL9727293 0.75 TP53 (0.59) GAATP53
SCHEMBL9727624 0.75 GAA (0.48) GAATP53AKR1C3MMP2
SCHEMBL25348950 0.74 MMP2 (0.62) GAATP53MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5164514-A Antispasmodics ROUSSEL UCLAF (FR) 1992-11-17 US disclosed
US-5081130-A Antispasmodic agents ROUSSEL UCLAF (FR) 1992-01-14 US disclosed
US-4990531-A Antispasmodic agents ROUSSEL UCLAF (FR) 1991-02-05 US disclosed
EP-0335758-A2 Derivatives of 1-arylsulfonyl-2-pyrolidinone, process for their preparation, their use as medicaments and compositions containing them ROUSSEL-UCLAF (FR) 1989-10-04 EP disclosed