SCHEMBL9727736

SCHEMBL9727736

COc1ccc(OCC=C(C)C)cc1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.48
MGAM O43451 3/20 0.48
GAA P10253 3/20 0.48
SI P14410 3/20 0.48
MGAM2 Q2M2H8 3/20 0.48
MTNR1A P48039 2/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
MAOB P27338 2/20 0.47
AOC3 Q16853 1/20 0.47
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46
MTNR1B P49286 1/20 0.44
PTPN1 P18031 1/20 0.44
ALOX5 P09917 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8036010 0.91 KDM4E (0.53) CYP19A1MGAMGAASIMGAM2
SCHEMBL4114408 0.85 KDM4E (0.49) MGAMGAASIMGAM2MTNR1A
SCHEMBL9856070 0.83 MGAM (0.55) MGAMGAASIMGAM2MTNR1A
SCHEMBL14012896 0.83 MAOB (0.52) GAAMTNR1AKDM4EALDH1A1MAOB
SCHEMBL20024720 0.82 MAPT (0.55) CYP19A1MTNR1AKDM4EALDH1A1MAOB
SCHEMBL670129 0.82 PPARD (0.49) GAAMTNR1AKDM4EALDH1A1MAOB
SCHEMBL9856624 0.82 KDM4E (0.46) CYP19A1MGAMGAASIMGAM2
SCHEMBL11555831 0.82 MAOB (0.53) GAAMTNR1AKDM4EALDH1A1MAOB
SCHEMBL791805 0.81 LMNA (0.53) MTNR1AKDM4EALDH1A1MAOBMTNR1B
SCHEMBL11269821 0.81 PPARG (0.44) MTNR1AALDH1A1MAOBAOC3MTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5091533-A Treating allergies, cardiovascular disorders, inflammation MERCK FROSST CANADA, INC. (CA) 1992-02-25 US disclosed
EP-0447189-A1 5-Hydroxy-2,3-dihydrobenzofuran analogs as leukotriene biosynthesis inhibitors MERCK FROSST CANADA INC. (CA) 1991-09-18 EP disclosed
US-4156725-A MICROBIOCIDES BURROUGHS WELLCOME CO. (US) 1979-05-29 US disclosed