SCHEMBL9728862

SCHEMBL9728862

Cc1nn2c(-c3cccc(C(F)(F)F)c3)ccnc2c1C(N)=O

nearest known ligand 0.69

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 10/20 0.69
PIM1 P11309 10/20 0.69
KDM4E B2RXH2 2/20 0.64
ACVR1 Q04771 2/20 0.60
CHEK1 O14757 3/20 0.52
CDK2 P24941 3/20 0.52
CSNK2A1 P68400 3/20 0.52
BRAF P15056 5/20 0.48
TLR8 Q9NR97 1/20 0.47
BTK Q06187 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11480970 0.87 BRAF (0.54) NTRK1PIM1KDM4EACVR1CHEK1
SCHEMBL9728647 0.82 KDM4E (0.48) NTRK1PIM1KDM4EACVR1CHEK1
SCHEMBL9878320 0.82 KDM4E (0.48) NTRK1PIM1KDM4EACVR1CHEK1
SCHEMBL3171563 0.80 KDM4E (0.54) NTRK1PIM1KDM4ECDK2BRAF
SCHEMBL11474283 0.78 KDM4E (0.60) NTRK1PIM1KDM4ECDK2BRAF
SCHEMBL11472391 0.78 NTRK1 (0.68) NTRK1PIM1KDM4EACVR1CDK2
SCHEMBL9728870 0.78 NTRK1 (0.65) NTRK1PIM1KDM4EACVR1CHEK1
SCHEMBL8435070 0.78 KDM4E (1.00) KDM4EBRAFTLR8
SCHEMBL11465926 0.78 BRAF (0.56) KDM4EBRAF
SCHEMBL11465978 0.77 KDM4E (0.52) NTRK1PIM1KDM4ECDK2BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5169850-A Neurotropic or hypotensive agents AMERICAN CYANAMID COMPANY (US) 1992-12-08 US disclosed
US-5059691-A Anxiolytic agents; hypotensive agents; nervous system disorders; cognition activators AMERICAN CYANAMID COMPANY (US) 1991-10-22 US disclosed