SCHEMBL9878320

SCHEMBL9878320

Cc1nn2c(-c3cccc(C(F)(F)F)c3)ccnc2c1C(=O)/N=C/N(C)C

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.48
NTRK1 P04629 6/20 0.47
PIM1 P11309 6/20 0.47
CHEK1 O14757 1/20 0.43
CDK2 P24941 1/20 0.43
CSNK2A1 P68400 1/20 0.43
BRAF P15056 10/20 0.42
ACVR1 Q04771 2/20 0.41
RAF1 P04049 1/20 0.40
MAPK14 Q16539 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9728647 1.00 KDM4E (0.48) KDM4ENTRK1PIM1CHEK1CDK2
SCHEMBL9877172 0.85 NTRK1 (0.64) KDM4ENTRK1PIM1CHEK1CDK2
SCHEMBL9728862 0.82 NTRK1 (0.69) KDM4ENTRK1PIM1CHEK1CDK2
SCHEMBL9877207 0.82 KDM4E (0.67) KDM4EBRAFRAF1MAPK14
SCHEMBL9728729 0.82 NTRK1 (0.53) KDM4ENTRK1PIM1CHEK1CDK2
SCHEMBL9877259 0.81 NTRK1 (0.43) NTRK1PIM1CHEK1CDK2CSNK2A1
SCHEMBL11480970 0.81 BRAF (0.54) KDM4ENTRK1PIM1CHEK1CDK2
SCHEMBL10842009 0.80 BRAF (0.45) KDM4EBRAF
SCHEMBL10842005 0.80 BRAF (0.45) KDM4EBRAF
SCHEMBL3171563 0.73 KDM4E (0.54) KDM4ENTRK1PIM1CDK2BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5059691-A Anxiolytic agents; hypotensive agents; nervous system disorders; cognition activators AMERICAN CYANAMID COMPANY (US) 1991-10-22 US claimed