SCHEMBL9728870

SCHEMBL9728870

Cc1nn2c(-c3ccccc3C(F)(F)F)ccnc2c1C(N)=O

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 10/20 0.65
PIM1 P11309 10/20 0.65
ACVR1 Q04771 2/20 0.57
CDK2 P24941 4/20 0.48
CHEK1 O14757 3/20 0.48
CSNK2A1 P68400 3/20 0.48
MAPT P10636 2/20 0.45
THRB P10828 1/20 0.45
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
SCN9A Q15858 3/20 0.41
SCN10A Q9Y5Y9 1/20 0.40
KMO O15229 1/20 0.39
CDC7 O00311 1/20 0.39
CCNE1 P24864 1/20 0.39
DBF4 Q9UBU7 1/20 0.39
NPFFR1 Q9GZQ6 1/20 0.38
NPFFR2 Q9Y5X5 1/20 0.38
BTK Q06187 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9877259 0.81 NTRK1 (0.43) NTRK1PIM1ACVR1CDK2CHEK1
SCHEMBL9728862 0.78 NTRK1 (0.69) NTRK1PIM1ACVR1CDK2CHEK1
SCHEMBL4307227 0.76 KMO (0.47) CDK2SCN9ASCN10AKMOCDC7
SCHEMBL9728834 0.74 NTRK1 (0.71) NTRK1PIM1ACVR1CDK2CHEK1
SCHEMBL11461808 0.73 KMO (0.41) CDK2SCN9ASCN10AKMOCDC7
SCHEMBL4307223 0.72 CDC7 (0.48) CDK2SCN9ASCN10AKMOCDC7
SCHEMBL27707931 0.71 SCN9A (0.44) CDK2MAPTSCN9ASCN10ACDC7
SCHEMBL31277907 0.70 NTRK1 (0.65) NTRK1PIM1ACVR1CDK2CHEK1
SCHEMBL11465849 0.70 BRAF (0.59) MAPTNPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL10941762 0.68 MAP2K1 (0.49) PIM1KMOKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5169850-A Neurotropic or hypotensive agents AMERICAN CYANAMID COMPANY (US) 1992-12-08 US disclosed
US-5059691-A Anxiolytic agents; hypotensive agents; nervous system disorders; cognition activators AMERICAN CYANAMID COMPANY (US) 1991-10-22 US disclosed