SCHEMBL9729180

SCHEMBL9729180

O=C1Cc2cccnc2C=C1Br

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.33
CDC25B P30305 1/20 0.33
BCHE P06276 1/20 0.33
TRIM24 O15164 1/20 0.32
TRIM33 Q9UPN9 1/20 0.32
CYP19A1 P11511 2/20 0.31
TNF P01375 2/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
TDP2 O95551 2/20 0.31
NSD2 O96028 2/20 0.31
PAX8 Q06710 2/20 0.31
ABL1 P00519 1/20 0.31
PLCG1 P19174 1/20 0.31
RIN1 Q13671 1/20 0.31
MEN1 O00255 1/20 0.31
THRB P10828 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9728723 0.76 TRIM24 (0.33) CES1BCHETRIM24TRIM33ALDH1A1
SCHEMBL12094093 0.71 HSP90AA1 (0.35) KDM4EALDH1A1TDP1
SCHEMBL30848588 0.69 KDM4E (0.33) KDM4EALDH1A1MEN1KMT2ATDP1
SCHEMBL2779620 0.68 GSK3A (0.39) CES1CDC25BCYP19A1TNFMAOA
SCHEMBL30482807 0.68 GSK3A (0.39) CES1CDC25BCYP19A1TNFMAOA
SCHEMBL1650021 0.68 KDM4E (0.40) MAOAMAOBKDM4EALDH1A1MEN1
SCHEMBL13859949 0.68 TSHR (0.35) CDC25BCYP19A1TNFMAOAMAOB
SCHEMBL30701903 0.67 CES1 (0.39) CES1CDC25BBCHEMAOAMAOB
SCHEMBL4964849 0.67 TRPA1 (0.32) CES1ALDH1A1TDP2NSD2PAX8
Hydrochloric Acid SCHEMBL30306200 0.67 KDM4E (0.39) MAOAMAOBKDM4EALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0250179-A2 BCD tricyclic ergoline part-structure analogues ELI LILLY AND COMPANY (US) 1987-12-23 EP claimed
US-5134143-A Dopamine Agonists ELI LILLY AND COMPANY (US) 1992-07-28 US disclosed
US-4977160-A DOPAMINE AGONISTS; PARKINSON*S DISEASE ELI LILLY AND COMPANY (US) 1990-12-11 US disclosed
US-4826986-A DOPAMINE AGONISTS ELI LILLY AND COMPANY (US) 1989-05-02 US disclosed
EP-0250179-A2 BCD tricyclic ergoline part-structure analogues ELI LILLY AND COMPANY (US) 1987-12-23 EP disclosed