SCHEMBL9729508

SCHEMBL9729508

CC1SC(=O)NN=C1c1ccc(N2CCNCC2)c(C#N)c1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 12/20 0.46
PDE3A Q14432 12/20 0.46
PDE4A P27815 5/20 0.46
PDE4B Q07343 5/20 0.46
PDE4C Q08493 5/20 0.46
PDE4D Q08499 5/20 0.46
KCNH2 Q12809 1/20 0.42
GPR119 Q8TDV5 1/20 0.41
BMPR1B O00238 2/20 0.39
BMPR1A P36894 2/20 0.39
ACVR1B P36896 2/20 0.39
ACVRL1 P37023 2/20 0.39
ACVR1 Q04771 2/20 0.39
FBP1 P09467 1/20 0.38
PIM1 P11309 1/20 0.37
CDK9 P50750 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7266588 0.83 GPR119 (0.59) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9729452 0.81 MAPT (0.45) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9039084 0.73 PDE3B (0.61) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL7273699 0.72 PDE3B (0.54) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL31116832 0.70 PDE3B (0.43) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9529826 0.69 PDE3B (0.70) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9729178 0.69 MAPT (0.46) PDE3BPDE3APDE4APDE4BPDE4C
Benzonitrile SCHEMBL9638199 0.69 PDE3B (0.58) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL3440910 0.69 PDE3B (0.62) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL7276709 0.68 GPR119 (0.62) PDE3BPDE3APDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5108998-A CARDIOTONIC THIADIAZINE DERIVATIVES HEUMANN PHARMA GMBH & CO. (DE) 1992-04-28 US disclosed