SCHEMBL9729772

SCHEMBL9729772

CN(C)CC=NC(=O)c1cnn2c(-c3cccnc3)ccnc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 1/20 0.47
CLK4 Q9HAZ1 1/20 0.47
DYRK1B Q9Y463 1/20 0.47
TLR8 Q9NR97 1/20 0.44
KDM4E B2RXH2 4/20 0.43
ALDH1A1 P00352 2/20 0.43
GAA P10253 2/20 0.43
LIMK1 P53667 2/20 0.43
MARK2 Q7KZI7 2/20 0.43
MAPK13 O15264 2/20 0.43
PIM1 P11309 4/20 0.41
MAPK9 P45984 1/20 0.41
DYRK1A Q13627 1/20 0.41
IRAK4 Q9NWZ3 1/20 0.41
GSK3A P49840 3/20 0.41
CDK1 P06493 1/20 0.41
MAPKAPK2 P49137 1/20 0.41
PLK1 P53350 1/20 0.41
AURKB Q96GD4 1/20 0.41
PDPK1 O15530 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9878097 0.81 MAP2K1 (0.49) MAP2K1CLK4DYRK1BTLR8KDM4E
SCHEMBL9878106 0.81 MAP2K1 (0.49) MAP2K1CLK4DYRK1BTLR8KDM4E
SCHEMBL11167079 0.78 MAP2K1 (0.59) MAP2K1CLK4DYRK1BTLR8KDM4E
SCHEMBL11162191 0.78 KDM4E (0.65) MAP2K1CLK4DYRK1BTLR8KDM4E
SCHEMBL11164960 0.77 BRAF (0.59) MAP2K1CLK4DYRK1BTLR8KDM4E
SCHEMBL9728973 0.77 CLK4 (0.61) MAP2K1CLK4DYRK1BTLR8KDM4E
SCHEMBL9728968 0.77 CLK4 (0.61) MAP2K1CLK4DYRK1BTLR8KDM4E
Hydrochloric Acid SCHEMBL11366478 0.77 KDM4E (0.64) MAP2K1CLK4DYRK1BTLR8KDM4E
SCHEMBL9728658 0.76 MAP2K1 (0.78) MAP2K1CLK4DYRK1BTLR8KDM4E
SCHEMBL11167453 0.75 MAP2K1 (0.57) MAP2K1CLK4DYRK1BTLR8KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5169850-A Neurotropic or hypotensive agents AMERICAN CYANAMID COMPANY (US) 1992-12-08 US disclosed
US-5059691-A Anxiolytic agents; hypotensive agents; nervous system disorders; cognition activators AMERICAN CYANAMID COMPANY (US) 1991-10-22 US disclosed