SCHEMBL9731535

SCHEMBL9731535

O=C(NC1CCCc2ccccc21)C(Cl)Cc1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.61
ALDH1A1 P00352 4/20 0.60
HTT P42858 2/20 0.57
EPHX2 P34913 2/20 0.57
MEN1 O00255 1/20 0.55
EPHX1 P07099 1/20 0.55
TAS1R3 Q7RTX0 5/20 0.54
TAS1R1 Q7RTX1 5/20 0.54
NPSR1 Q6W5P4 1/20 0.54
TAS1R2 Q8TE23 3/20 0.53
SMN1; SMN2 Q16637 1/20 0.52
HPGD P15428 1/20 0.52
TSHR P16473 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29131632 0.85 OPRK1 (0.59) KMT2AALDH1A1HTTEPHX2MEN1
SCHEMBL29131630 0.85 OPRK1 (0.59) KMT2AALDH1A1HTTEPHX2MEN1
SCHEMBL54832 0.81 HTT (0.61) KMT2AALDH1A1HTTMEN1EPHX1
SCHEMBL29131636 0.81 KMT2A (0.54) KMT2AALDH1A1HTTEPHX2MEN1
SCHEMBL29131637 0.81 KMT2A (0.54) KMT2AALDH1A1HTTEPHX2MEN1
SCHEMBL9731131 0.79 ALDH1A1 (0.75) KMT2AALDH1A1HTTEPHX2MEN1
SCHEMBL5651521 0.79 TAOK3 (0.58) KMT2AALDH1A1HTTEPHX2MEN1
SCHEMBL29131614 0.79 EPHX2 (0.60) KMT2AALDH1A1HTTEPHX2MEN1
SCHEMBL29131610 0.79 EPHX2 (0.60) KMT2AALDH1A1HTTEPHX2MEN1
SCHEMBL18351574 0.78 TAOK1 (0.57) KMT2AALDH1A1HTTMEN1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5151446-A Neurological disorders or cardiovascular disorders NORTHWESTERN UNIVERSITY (US) 1992-09-29 US disclosed
US-5071875-A Nervous system, psychological disorders; sleep cycle, skin dis coloration NORTHWESTERN UNIVERSITY (US) 1991-12-10 US disclosed
EP-0420064-A2 Substituted 2-amidotetralins as melatonin agonists and antagonists NORTHWESTERN UNIVERSITY (US) 1991-04-03 EP disclosed