SCHEMBL9733150

SCHEMBL9733150

O=[N+]([O-])c1ccc2nc(C3CNCCN3)ccc2c1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.51
HTR3E A5X5Y0 1/20 0.51
HTR3B O95264 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
SLC6A4 P31645 1/20 0.51
CYP2C19 P33261 1/20 0.51
THPO P40225 1/20 0.51
HTR3A P46098 1/20 0.51
HTR3D Q70Z44 1/20 0.51
HTR3C Q8WXA8 1/20 0.51
LMNA P02545 1/20 0.44
PMP22 Q01453 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
TTR P02766 1/20 0.37
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3856968 0.82 ALDH1A1 (0.48) ALDH1A1HTR3EHTR3BCYP1A2CYP3A4
SCHEMBL9318637 0.80 TYMS (0.38) ALDH1A1HTR3EHTR3BCYP1A2CYP3A4
SCHEMBL9318307 0.80 NQO2 (0.40) ALDH1A1HTR3EHTR3BCYP1A2CYP3A4
SCHEMBL9318047 0.80 ALDH1A1 (0.43) ALDH1A1HTR3EHTR3BCYP1A2CYP3A4
SCHEMBL6699333 0.78 MAPT (0.39) ALDH1A1CYP1A2LMNANPSR1
SCHEMBL28752901 0.78 HRH3 (0.37) HTR3EHTR3BSLC6A4HTR3AHTR3D
SCHEMBL27627374 0.78 BACE1 (0.41)
SCHEMBL27608178 0.78 BACE1 (0.41) SLC6A4
SCHEMBL31458446 0.76 ALDH1A1 (0.50) ALDH1A1HTR3EHTR3BCYP1A2CYP3A4
SCHEMBL9319076 0.75 ALDH1A1 (0.31) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-3199969-A None JP disclosed
CN-101239953-A Antidepressant arylpiperazine derivatives of heterocycle-fused benzodioxans WYETH CORP (US) 2008-08-13 CN disclosed
CN-100340562-C Antidepressant arylpiperazine derivatives of heterocycle-fused benzodioxans WYETH CORP (US) 2007-10-03 CN disclosed
CN-1681822-A Antidepressant arylpiperazine derivatives of heterocycle-fused benzodioxans WYETH CORP (US) 2005-10-12 CN disclosed
US-5120641-A Incubating with sample, determining radioactivity DAIICHI PURE CHEMICALS CO., LTD. (JP) 1992-06-09 US disclosed
JP-H03199969-A METHOD FOR MEASURING RETAKING PART OF SEROTONIN AND RADIO LIGAND USED IN THIS METHOD DAI ICHI PURE CHEM CO LTD 1991-08-30 JP disclosed
EP-0435192-A2 Method for measurement of serotonin uptake sites and radioligand therefor DAIICHI PURE CHEMICALS CO. LTD. (JP) 1991-07-03 EP disclosed