SCHEMBL9733733

SCHEMBL9733733

COC(=O)C(C)C(=O)Cc1ccc(OC)cc1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.57
ALDH1A1 P00352 3/20 0.50
KLK7 P49862 3/20 0.50
KDM4E B2RXH2 1/20 0.49
POLB P06746 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
LDHA P00338 1/20 0.49
CNR2 P34972 1/20 0.48
NPC1 O15118 1/20 0.48
PKM P14618 1/20 0.48
LMNA P02545 1/20 0.48
CTBP2 P56545 1/20 0.47
F2RL1 P55085 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9734555 0.85 ESR1 (0.53) HTTSMN1; SMN2LMNA
SCHEMBL28657956 0.85 LDHA (0.59) HTTALDH1A1KLK7KDM4EPOLB
SCHEMBL9780185 0.83 HTT (0.38) HTTALDH1A1KLK7POLB
SCHEMBL3829820 0.82 HTT (0.59) HTTALDH1A1KLK7KDM4EPOLB
SCHEMBL9780186 0.81 SLC6A4 (0.46) ALDH1A1KDM4ELMNA
SCHEMBL27985109 0.80 ALDH1A1 (0.55) HTTALDH1A1POLBSMN1; SMN2LDHA
SCHEMBL28500649 0.79 HTT (0.56) HTTALDH1A1KLK7KDM4EPOLB
SCHEMBL8951701 0.79 HTT (0.56) HTTALDH1A1KLK7SMN1; SMN2LDHA
SCHEMBL27746899 0.79 HTT (0.59) HTTALDH1A1KDM4EPOLBSMN1; SMN2
SCHEMBL11082660 0.77 HTT (0.58) HTTALDH1A1KDM4EPOLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5135940-A Antiallegens, antiinflammatory agents MERCK FROSST CANADA, INC. (CA) 1992-08-04 US disclosed
EP-0252639-A1 Leukotriene antagonists MERCK FROSST CANADA INC. (CA) 1988-01-13 EP disclosed
EP-0104885-B1 LEUKOTRIENE ANTAGONISTS, THEIR PRODUCTION, AND COMPOSITIONS CONTAINING THEM MERCK FROSST CANADA INC. (CA) 1986-06-04 EP disclosed
EP-0156233-A2 Use of leukotriene antagonists for producing cytoprotective pharmaceutical compositions and process for producing cytoprotective pharmaceutical compositions MERCK & CO. INC. (US) 1985-10-02 EP disclosed
EP-0104885-A1 Leukotriene antagonists, their production, and compositions containing them MERCK FROSST CANADA INC. (CA) 1984-04-04 EP disclosed