SCHEMBL9733876

SCHEMBL9733876

c1ccc(-c2ccnc(CN3CCCC3)c2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 1/20 0.47
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 2/20 0.47
CXCR4 P61073 1/20 0.47
HPGD P15428 1/20 0.47
HSD17B10 Q99714 1/20 0.47
LTA4H P09960 2/20 0.47
TSHR P16473 2/20 0.46
MAPT P10636 1/20 0.46
MAPK1 P28482 1/20 0.46
BACE1 P56817 1/20 0.46
CYP2D6 P10635 1/20 0.45
CYP2C19 P33261 1/20 0.45
HCRTR1 O43613 1/20 0.44
HCRTR2 O43614 1/20 0.44
KDM5C P41229 1/20 0.43
KDM4C Q9H3R0 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
KDR P35968 1/20 0.43
DRD2 P14416 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13940646 0.89 KMT2A (0.45) TMEM97ALDH1A1KDM4ECXCR4TSHR
SCHEMBL7498479 0.85 DRD4 (0.59) ALDH1A1KDM4ETSHRMAPTDRD2
SCHEMBL30484462 0.84 EGLN1 (0.47) ALDH1A1KDM4ETSHRMAPTMAPK1
SCHEMBL29204511 0.84 EGLN1 (0.46) ALDH1A1KDM4ETSHRMAPTMAPK1
SCHEMBL7500264 0.84 ALDH1A1 (0.66) ALDH1A1KDM4EHSD17B10TSHRDRD2
SCHEMBL30484482 0.83 EGLN1 (0.46) ALDH1A1KDM4ETSHRMAPTMAPK1
SCHEMBL10375167 0.83 TRPV6 (0.53) ALDH1A1KDM4ESIGMAR1DRD2DRD4
SCHEMBL29204494 0.83 HRH3 (0.51) ALDH1A1KDM4ETSHRMAPTMAPK1
SCHEMBL29204460 0.83 EGLN1 (0.48) ALDH1A1KDM4ETSHRMAPTMAPK1
SCHEMBL29204466 0.83 EGLN1 (0.48) ALDH1A1KDM4ETSHRMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5114945-A Spiropiperidine derivatives GLAXO GROUP LIMITED (GB) 1992-05-19 US disclosed
EP-0330461-A2 Piperidine derivatives GLAXO GROUP LIMITED (GB) 1989-08-30 EP disclosed