SCHEMBL9733974

SCHEMBL9733974

CCC(=O)c1ccc(SC)cc1Br

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
KMT2A Q03164 4/20 0.44
MEN1 O00255 3/20 0.44
HSP90AB1 P08238 1/20 0.43
MCL1 Q07820 1/20 0.42
HPGD P15428 5/20 0.41
POLB P06746 2/20 0.41
HSD17B10 Q99714 3/20 0.40
ADORA3 P0DMS8 2/20 0.39
ADORA2A P29274 1/20 0.39
ADORA2B P29275 1/20 0.39
ADORA1 P30542 1/20 0.39
GAA P10253 2/20 0.38
TSHR P16473 3/20 0.37
HTT P42858 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
NPC1 O15118 1/20 0.36
MITF O75030 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31229283 0.81 ALDH1A1 (0.45) ALDH1A1KMT2AMEN1HSP90AB1MCL1
SCHEMBL21951012 0.81 ALDH1A1 (0.65) ALDH1A1KMT2AMEN1HSP90AB1MCL1
SCHEMBL2257900 0.81 ALDH1A1 (0.45) ALDH1A1KMT2AMEN1HSP90AB1MCL1
SCHEMBL12726114 0.80 MCL1 (0.46) ALDH1A1KMT2AMCL1HPGDPOLB
SCHEMBL10274092 0.80 MCL1 (0.59) ALDH1A1KMT2AMEN1MCL1HPGD
SCHEMBL5678085 0.79 ALDH1A1 (0.44) ALDH1A1KMT2AMEN1HSP90AB1MCL1
SCHEMBL9560116 0.79 ALDH1A1 (0.44) ALDH1A1KMT2AMEN1HSP90AB1MCL1
SCHEMBL11310587 0.79 ALDH1A1 (0.39) ALDH1A1HSP90AB1HPGDPOLBHSD17B10
SCHEMBL6174178 0.78 HSP90AB1 (0.48) ALDH1A1KMT2AHSP90AB1HPGDPOLB
SCHEMBL4766604 0.78 ALDH1A1 (0.43) ALDH1A1KMT2AMEN1MCL1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5135940-A Antiallegens, antiinflammatory agents MERCK FROSST CANADA, INC. (CA) 1992-08-04 US disclosed
EP-0252639-A1 Leukotriene antagonists MERCK FROSST CANADA INC. (CA) 1988-01-13 EP disclosed