SCHEMBL9734648

SCHEMBL9734648

CCn1c(=O)n(C)c(=O)c2c(-c3ccc(F)cc3)c(C=CC=O)c(C(C)C)nc21

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.42
GCGR P47871 4/20 0.38
HTT P42858 1/20 0.36
NCOA3 Q9Y6Q9 1/20 0.36
MAPK1 P28482 1/20 0.34
GFER P55789 1/20 0.34
HMGCR P04035 2/20 0.33
MAPK14 Q16539 1/20 0.33
ESR1 P03372 1/20 0.33
CHRM1 P11229 1/20 0.33
TBXA2R P21731 1/20 0.33
PDE4A P27815 1/20 0.33
ADRA1A P35348 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9387195 1.00 DPP4 (0.42) DPP4GCGRHTTNCOA3MAPK1
SCHEMBL9735873 0.84 DPP4 (0.41) DPP4HTTNCOA3HMGCRMAPK14
SCHEMBL9735875 0.84 DPP4 (0.41) DPP4HTTNCOA3HMGCRMAPK14
SCHEMBL9384186 0.83 GCGR (0.38) GCGRMAPK1HMGCRESR1CHRM1
SCHEMBL9735137 0.83 GCGR (0.38) GCGRMAPK1HMGCRESR1CHRM1
SCHEMBL9736971 0.80 HMGCR (0.60) HMGCR
SCHEMBL9383849 0.80 HMGCR (0.60) HMGCR
SCHEMBL9383855 0.80 HMGCR (0.60) HMGCR
SCHEMBL9736966 0.80 HMGCR (0.60) HMGCR
SCHEMBL9383858 0.80 HMGCR (0.60) HMGCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5145959-A Enzyme inhibitors; antilipemic agents; treatment of atherosclerosis BAYER AKTIENGESELLSCHAFT (DE) 1992-09-08 US disclosed
US-5075311-A Anticholesterol agents BAYER AKTIENGESELLSCHAFT (DE) 1991-12-24 US disclosed