SCHEMBL9735137

SCHEMBL9735137

CCn1c(=O)[nH]c(=O)c2c(-c3ccc(F)cc3)c(C=CC=O)c(C(C)C)nc21

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GCGR P47871 5/20 0.38
RXFP1 Q9HBX9 2/20 0.37
TPH1 P17752 2/20 0.35
TPH2 Q8IWU9 2/20 0.35
KDM4E B2RXH2 4/20 0.34
MAPK1 P28482 2/20 0.33
ALDH1A1 P00352 2/20 0.33
HMGCR P04035 2/20 0.33
ESR1 P03372 1/20 0.33
CHRM1 P11229 1/20 0.33
TBXA2R P21731 1/20 0.33
PDE4A P27815 1/20 0.33
ADRA1A P35348 1/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9384186 1.00 GCGR (0.38) GCGRRXFP1TPH1TPH2KDM4E
SCHEMBL9388048 0.91 KDM4E (0.45) GCGRRXFP1KDM4EMAPK1ALDH1A1
SCHEMBL9736896 0.91 KDM4E (0.45) GCGRRXFP1KDM4EMAPK1ALDH1A1
SCHEMBL9736194 0.90 GCGR (0.40) GCGRRXFP1TPH1TPH2KDM4E
SCHEMBL9736133 0.87 GCGR (0.37) GCGRALDH1A1TP53
SCHEMBL9736123 0.87 GCGR (0.37) GCGRALDH1A1TP53
SCHEMBL9736090 0.84 RXRA (0.40) RXFP1TPH1TPH2KDM4EMAPK1
SCHEMBL9384462 0.84 RXRA (0.40) RXFP1TPH1TPH2KDM4EMAPK1
SCHEMBL9734648 0.83 DPP4 (0.42) GCGRMAPK1HMGCRESR1CHRM1
SCHEMBL9387195 0.83 DPP4 (0.42) GCGRMAPK1HMGCRESR1CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5145959-A Enzyme inhibitors; antilipemic agents; treatment of atherosclerosis BAYER AKTIENGESELLSCHAFT (DE) 1992-09-08 US disclosed
US-5075311-A Anticholesterol agents BAYER AKTIENGESELLSCHAFT (DE) 1991-12-24 US disclosed