SCHEMBL9735142

SCHEMBL9735142

CC(C)c1nc2[nH]c(=O)[nH]c(=O)c2c(-c2ccc(F)cc2)c1C=CC(O)CC(=O)CC(=O)O

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 4/20 0.49
ESR1 P03372 1/20 0.49
CHRM1 P11229 1/20 0.49
TBXA2R P21731 1/20 0.49
PDE4A P27815 1/20 0.49
ADRA1A P35348 1/20 0.49
ALDH1A1 P00352 1/20 0.42
CYP3A4 P08684 1/20 0.42
PDE6D O43924 1/20 0.42
NR1I2 O75469 1/20 0.42
PDE4D Q08499 1/20 0.42
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
ABCC3 O15438 1/20 0.38
ABCC4 O15439 1/20 0.38
GCGR P47871 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9735125 1.00 HMGCR (0.49) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL9387121 0.92 HMGCR (0.47) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL9735282 0.84 HMGCR (0.57) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL9734698 0.81 HMGCR (0.43) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL9734676 0.81 HMGCR (0.43) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL9482432 0.79 HMGCR (0.56) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL9482422 0.79 HMGCR (0.56) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL9735571 0.79 GCGR (0.39) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL9383069 0.79 GCGR (0.39) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL9382441 0.78 GCGR (0.42) HMGCRALDH1A1GCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5145959-A Enzyme inhibitors; antilipemic agents; treatment of atherosclerosis BAYER AKTIENGESELLSCHAFT (DE) 1992-09-08 US disclosed
US-5075311-A Anticholesterol agents BAYER AKTIENGESELLSCHAFT (DE) 1991-12-24 US disclosed