SCHEMBL9735571

SCHEMBL9735571

CC(C)c1nc2[nH]c(=O)[nH]c(=O)c2c(-c2ccc(F)cc2)c1C=CC=O

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GCGR P47871 3/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38
TYMP P19971 1/20 0.37
IDO1 P14902 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ALDH1A1 P00352 1/20 0.35
HMGCR P04035 5/20 0.34
ESR1 P03372 1/20 0.34
CHRM1 P11229 1/20 0.34
TBXA2R P21731 1/20 0.34
PDE4A P27815 1/20 0.34
ADRA1A P35348 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9383069 1.00 GCGR (0.39) GCGRCYP1A2CYP2C19TYMPIDO1
SCHEMBL9382441 0.89 GCGR (0.42) GCGRCYP1A2CYP2C19TYMPIDO1
SCHEMBL9736123 0.81 GCGR (0.37) GCGRCYP1A2CYP2C19IDO1ALDH1A1
SCHEMBL9736133 0.81 GCGR (0.37) GCGRCYP1A2CYP2C19IDO1ALDH1A1
SCHEMBL8949683 0.80 GCGR (0.53) GCGRHMGCRESR1CHRM1TBXA2R
SCHEMBL9523672 0.80 GCGR (0.40) GCGRCYP1A2CYP2C19HMGCRESR1
SCHEMBL9791356 0.80 GCGR (0.40) GCGRCYP1A2CYP2C19HMGCRESR1
SCHEMBL9735142 0.79 HMGCR (0.49) GCGRALDH1A1HMGCRESR1CHRM1
SCHEMBL9735125 0.79 HMGCR (0.49) GCGRALDH1A1HMGCRESR1CHRM1
SCHEMBL9384186 0.78 GCGR (0.38) GCGRALDH1A1HMGCRESR1CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5145959-A Enzyme inhibitors; antilipemic agents; treatment of atherosclerosis BAYER AKTIENGESELLSCHAFT (DE) 1992-09-08 US disclosed
US-5075311-A Anticholesterol agents BAYER AKTIENGESELLSCHAFT (DE) 1991-12-24 US disclosed