SCHEMBL9735224

SCHEMBL9735224

Cn1nc(SC2c3cc(C#N)ccc3CC(C)(C)C2O)ccc1=O

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 5/20 0.36
ABCC9 O60706 9/20 0.35
ABCC8 Q09428 2/20 0.35
KCNJ11 Q14654 2/20 0.35
KCNJ8 Q15842 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
LMNA P02545 1/20 0.35
CNR2 P34972 1/20 0.35
ABCB1 P08183 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9738782 0.81 CNR2 (0.37) BACE1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL9733745 0.78 ABCC9 (0.38) ABCC9CNR2ABCB1
SCHEMBL9733386 0.73 ABCC9 (0.37) BACE1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL9734096 0.70 ABCC9 (0.41) BACE1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL1573018 0.69 CYP11B1 (0.49) ABCC9ABCC8KCNJ11KCNJ8CYP1A2
SCHEMBL10560531 0.68 CNR2 (0.42) BACE1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL10560535 0.68 CNR2 (0.42) BACE1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL9733193 0.68 ABCC9 (0.38) BACE1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL9472527 0.67 ABCB1 (0.35) BACE1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL9733302 0.67 ABCC9 (0.38) BACE1ABCC9ABCC8KCNJ11KCNJ8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132307-A TETRALIN COMPOUNDS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-07-21 US disclosed
EP-0368160-A1 Tetralin derivatives MERCK PATENT GmbH (DE) 1990-05-16 EP disclosed