SCHEMBL9735829

SCHEMBL9735829

CC1(CNC(=O)OCc2ccccc2)Cc2ccc(C#N)cc2C(n2ccccc2=O)O1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADAM10 O14672 1/20 0.38
MMP2 P08253 1/20 0.38
MMP9 P14780 1/20 0.38
MMP14 P50281 1/20 0.38
ADAM17 P78536 1/20 0.38
CYP3A4 P08684 1/20 0.37
ALOX15 P16050 1/20 0.37
PREP P48147 2/20 0.37
ABCB1 P08183 6/20 0.36
CTSL P07711 4/20 0.35
CTSB P07858 3/20 0.35
CTSK P43235 2/20 0.35
GAA P10253 1/20 0.35
CTSS P25774 3/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9198396 0.82 ABCC9 (0.39) ABCB1
SCHEMBL9197783 0.80 ABCB1 (0.34) ABCB1
SCHEMBL9735028 0.80 ABCC9 (0.37) ABCB1
SCHEMBL9737142 0.71 MAOB (0.42) CYP3A4ALOX15ABCB1CTSLCTSB
SCHEMBL9734265 0.69 ABCC9 (0.39) CYP3A4ALOX15ABCB1
SCHEMBL9734096 0.68 ABCC9 (0.41) CYP3A4ABCB1
SCHEMBL9735833 0.68 CYP3A4 (0.38) ADAM10MMP2MMP9MMP14ADAM17
SCHEMBL9198634 0.68 ABCC9 (0.34) ABCB1
SCHEMBL9733575 0.67 ABCC9 (0.37) ABCB1
SCHEMBL9736930 0.67 MEN1 (0.32) GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5130322-A CHROMAN DERIVATIVES MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-07-14 US disclosed
EP-0415065-A1 Chroman derivatives MERCK PATENT GmbH (DE) 1991-03-06 EP disclosed