SCHEMBL9735945

SCHEMBL9735945

CC1(COC2CCCCO2)C=Cc2cc(C#N)ccc2O1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
XDH P47989 1/20 0.36
CHEK1 O14757 3/20 0.35
ABCB1 P08183 8/20 0.34
HIF1A Q16665 2/20 0.33
EPAS1 Q99814 2/20 0.33
KDM4C Q9H3R0 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
CA12 O43570 1/20 0.32
CA9 Q16790 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9736524 0.78 PTGS1 (0.46) PTGS1PTGS2XDHABCB1CA12
SCHEMBL9736544 0.74 ABCB1 (0.41) ABCB1
SCHEMBL9274003 0.74 MAOB (0.37) CHEK1ABCB1MEN1KMT2A
SCHEMBL22939295 0.69 BACE1 (0.32) ABCB1MEN1KMT2A
SCHEMBL506743 0.68 CA12 (0.46) PTGS1PTGS2XDHABCB1HIF1A
SCHEMBL30523681 0.68 CA12 (0.46) PTGS1PTGS2XDHABCB1HIF1A
SCHEMBL9736953 0.67 ABCB1 (0.38) ABCB1
SCHEMBL15633452 0.67 KDM4C (0.39) CHEK1KDM4CNPC1RAB9AMEN1
SCHEMBL8534981 0.67 CA12 (0.40) PTGS1PTGS2XDHABCB1HIF1A
SCHEMBL5857069 0.66 TACR1 (0.45) KDM4CNPC1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5130322-A CHROMAN DERIVATIVES MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-07-14 US disclosed