SCHEMBL9735954

SCHEMBL9735954

CCc1ccc2c(c1)cc1n2CCC1NO

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 7/20 0.35
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
S1PR5 Q9H228 2/20 0.33
S1PR4 O95977 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2A6 P11509 1/20 0.33
HDAC8 Q9BY41 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9735960 0.75 S1PR1 (0.36) S1PR1S1PR5
SCHEMBL26433370 0.65 HTR2A (0.43) ALDH1A1ALOX15CYP1A2CYP2A6
SCHEMBL9736283 0.63 SRD5A1 (0.40) KDM4EALDH1A1HPGDNPC1RAB9A
SCHEMBL21871188 0.61 GPR119 (0.49) CYP1A2CYP2A6HDAC8
SCHEMBL30703015 0.59 HTR2A (0.43) S1PR1
SCHEMBL16979076 0.58 CYP1A2 (0.44) KDM4EALDH1A1HPGDALOX15CYP1A2
SCHEMBL29407167 0.57 CYP2A6 (0.80) ALDH1A1NPC1RAB9ACYP1A2CYP2A6
SCHEMBL347592 0.57 CYP2A6 (0.80) ALDH1A1NPC1RAB9ACYP1A2CYP2A6
SCHEMBL9613258 0.56 HSD17B10 (0.62) KDM4EALDH1A1HPGDALOX15CYP1A2
SCHEMBL27547839 0.56 CYP1A2 (0.61) ALDH1A1NPC1RAB9ACYP1A2CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992021678-A1 LIPOXYGENASE INHIBITING PYRROLO [1,2a]INDOLE COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1992-12-10 WO disclosed