SCHEMBL9735960

SCHEMBL9735960

CCc1ccc2c(c1)cc1n2CCC1N(O)C(N)=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 8/20 0.36
S1PR5 Q9H228 1/20 0.33
AKR1C3 P42330 1/20 0.33
AKR1C2 P52895 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9737528 0.76 GALR3 (0.42)
SCHEMBL9735954 0.75 S1PR1 (0.35) S1PR1S1PR5
SCHEMBL9613272 0.62 TP53 (0.47) AKR1C3AKR1C2
SCHEMBL9736283 0.61 SRD5A1 (0.40) AKR1C3AKR1C2
SCHEMBL9613258 0.57 HSD17B10 (0.62) AKR1C3AKR1C2
SCHEMBL12125696 0.56 LCK (0.56) AKR1C3AKR1C2
SCHEMBL806188 0.56 NOTUM (0.54) S1PR1AKR1C3AKR1C2
SCHEMBL30703015 0.55 HTR2A (0.43) S1PR1
SCHEMBL20921201 0.55 MEN1 (0.46) AKR1C3AKR1C2
Acetamide SCHEMBL27414047 0.54 ALDH1A1 (0.58)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992021678-A1 LIPOXYGENASE INHIBITING PYRROLO [1,2a]INDOLE COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1992-12-10 WO disclosed