SCHEMBL9737641

SCHEMBL9737641

O=CC(F)(F)[C@H](OOCOCc1ccccc1)[C@H](O)COOCOCc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.38
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
TSHR P16473 2/20 0.35
TACR1 P25103 2/20 0.34
MAPK1 P28482 1/20 0.33
KMT2A Q03164 1/20 0.33
HTT P42858 2/20 0.33
AR P10275 1/20 0.33
PTPN1 P18031 1/20 0.33
SLC1A1 P43005 1/20 0.32
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32
CYP3A4 P08684 1/20 0.32
ALOX15 P16050 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
BACE1 P56817 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9737400 1.00 CA1 (0.38) CA1CA2CA7CA9TSHR
SCHEMBL9736749 0.88 CA1 (0.35) CA1CA2CA7CA9TSHR
SCHEMBL9735971 0.88 CA1 (0.35) CA1CA2CA7CA9TSHR
SCHEMBL9737639 0.77 PTPN1 (0.37) TSHRMAPK1KMT2APTPN1SMN1; SMN2
SCHEMBL9770003 0.77 PTPN1 (0.37) TSHRMAPK1KMT2APTPN1SMN1; SMN2
SCHEMBL2117279 0.65 CA1 (0.44) CA1CA2CA7CA9TSHR
SCHEMBL29425704 0.64 CA1 (0.47) CA1CA2CA7CA9TSHR
SCHEMBL30712001 0.64 CA1 (0.47) CA1CA2CA7CA9TSHR
SCHEMBL6832294 0.64 TSHR (0.64) CA1CA2CA7CA9TSHR
SCHEMBL4483094 0.63 CA1 (0.53) CA1CA2CA7CA9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5118820-A Carbohydrate is chemical intermediate for nucleoside ELI LILLY AND COMPANY (US) 1992-06-02 US disclosed
US-5015743-A 2-Deoxy-2,2-difluororibose ELI LILLY AND COMPANY (US) 1991-05-14 US disclosed
US-4808614-A Difluoro antivirals and intermediate therefor ELI LILLY AND COMPANY (US) 1989-02-28 US disclosed
EP-0122707-B1 IMPROVEMENTS IN OR RELATING TO NOVEL DIFLUORO ANTIVIRAL AGENTS ELI LILLY AND COMPANY (US) 1987-09-16 EP disclosed
US-4692434-A NUCLEOSIDES ELI LILLY AND COMPANY (US) 1987-09-08 US disclosed
EP-0211354-A2 Nucleosides and their use as antineoplastic agents MERRELL DOW PHARMACEUTICALS INC. (US) 1987-02-25 EP disclosed
US-4526988-A Hydrolyzing alkyl 3-dioxolanyl-2,2-difluoro-3-hydroxy propionate ELI LILLY AND COMPANY (US) 1985-07-02 US disclosed
EP-0122707-A1 Improvements in or relating to novel difluoro antiviral agents ELI LILLY AND COMPANY (US) 1984-10-24 EP disclosed