SCHEMBL9736749

SCHEMBL9736749

O=CC(F)(F)[C@H](OOCc1ccccc1)[C@@H](O)COOCc1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.35
PTPN1 P18031 3/20 0.35
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
PTPRC P08575 1/20 0.33
TSHR P16473 1/20 0.33
TACR1 P25103 1/20 0.32
SLC1A3 P43003 2/20 0.32
SLC1A2 P43004 2/20 0.32
SLC1A1 P43005 2/20 0.32
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
CYP3A4 P08684 1/20 0.32
ALOX15 P16050 1/20 0.32
BACE1 P56817 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9735971 1.00 CA1 (0.35) CA1PTPN1CA2CA7CA9
SCHEMBL9737641 0.88 CA1 (0.38) CA1PTPN1CA2CA7CA9
SCHEMBL9737400 0.88 CA1 (0.38) CA1PTPN1CA2CA7CA9
SCHEMBL9770003 0.81 PTPN1 (0.37) PTPN1PTPRCTSHRKMT2AMEN1
SCHEMBL9737639 0.81 PTPN1 (0.37) PTPN1PTPRCTSHRKMT2AMEN1
SCHEMBL8992078 0.69 SLC1A1 (0.41) CA1CA2CA7CA9SLC1A3
SCHEMBL4412607 0.69 CA1 (0.43) CA1CA2CA7CA9TSHR
SCHEMBL620071 0.68 CA1 (0.53) CA1CA2CA7CA9TSHR
SCHEMBL4411606 0.66 CA1 (0.41) CA1CA2CA7CA9TSHR
SCHEMBL4409725 0.66 CA1 (0.41) CA1CA2CA7CA9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5118820-A Carbohydrate is chemical intermediate for nucleoside ELI LILLY AND COMPANY (US) 1992-06-02 US disclosed
US-5015743-A 2-Deoxy-2,2-difluororibose ELI LILLY AND COMPANY (US) 1991-05-14 US disclosed
US-4808614-A Difluoro antivirals and intermediate therefor ELI LILLY AND COMPANY (US) 1989-02-28 US disclosed
EP-0122707-B1 IMPROVEMENTS IN OR RELATING TO NOVEL DIFLUORO ANTIVIRAL AGENTS ELI LILLY AND COMPANY (US) 1987-09-16 EP disclosed
US-4692434-A NUCLEOSIDES ELI LILLY AND COMPANY (US) 1987-09-08 US disclosed
EP-0211354-A2 Nucleosides and their use as antineoplastic agents MERRELL DOW PHARMACEUTICALS INC. (US) 1987-02-25 EP disclosed
US-4526988-A Hydrolyzing alkyl 3-dioxolanyl-2,2-difluoro-3-hydroxy propionate ELI LILLY AND COMPANY (US) 1985-07-02 US disclosed
EP-0122707-A1 Improvements in or relating to novel difluoro antiviral agents ELI LILLY AND COMPANY (US) 1984-10-24 EP disclosed