SCHEMBL9738251

SCHEMBL9738251

C=CCOC(=O)N1C[C@@H](SCc2ccc(OC)cc2)C[C@H]1C=C(C)C(N)=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTRA1 Q92743 1/20 0.36
ALDH1A1 P00352 3/20 0.34
DPP4 P27487 3/20 0.34
DPP7 Q9UHL4 3/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2D6 P10635 1/20 0.34
MAPT P10636 1/20 0.34
CYP2C19 P33261 1/20 0.34
MAPKAPK2 P49137 1/20 0.34
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
TP53 P04637 2/20 0.33
TSHR P16473 2/20 0.33
FAP Q12884 2/20 0.33
DPP8 Q6V1X1 2/20 0.33
DPP9 Q86TI2 2/20 0.33
CYP19A1 P11511 1/20 0.33
HPGD P15428 1/20 0.32
IDO1 P14902 2/20 0.32
ALOX15 P16050 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9738245 1.00 HTRA1 (0.36) HTRA1ALDH1A1DPP4DPP7CYP3A4
SCHEMBL9738733 0.88 HTRA1 (0.38) HTRA1ALDH1A1DPP4DPP7CYP3A4
SCHEMBL9737498 0.82 CYP19A1 (0.42) HTRA1ALDH1A1DPP4DPP7CYP3A4
SCHEMBL9738363 0.81 HTRA1 (0.37) HTRA1ALDH1A1DPP4DPP7CYP3A4
SCHEMBL9737552 0.73 SIGMAR1 (0.33) CYP19A1SIGMAR1
SCHEMBL9737546 0.73 SIGMAR1 (0.33) CYP19A1SIGMAR1
SCHEMBL5414235 0.73 DPP4 (0.43) HTRA1ALDH1A1DPP4DPP7MAPT
SCHEMBL8545366 0.72 FABP7 (0.36) ALDH1A1MAPKAPK2CA1CA2TP53
SCHEMBL8095363 0.70 GAA (0.44) ALDH1A1MAPTSMN1; SMN2
SCHEMBL9202402 0.70 HTRA1 (0.44) HTRA1ALDH1A1DPP4DPP7MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5095013-A Antibiotics BANYU PHARMACEUTICAL CO., LTD. (JP) 1992-03-10 US disclosed
EP-0411664-A2 2-(2-Vinylpyrrolidinylthio)carbapenem derivatives Banyu Pharmaceutical Co., Ltd. (JP) 1991-02-06 EP disclosed