SCHEMBL9738860

SCHEMBL9738860

O=C1c2ccc(Sc3ccccc3)cc2C(=O)c2cc3ccccc3cc21

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCL2 P10415 5/20 0.73
MCL1 Q07820 5/20 0.73
MAOA P21397 4/20 0.57
MAOB P27338 4/20 0.57
ADORA2A P29274 1/20 0.44
MAPT P10636 3/20 0.42
MAPK1 P28482 2/20 0.42
KDM4E B2RXH2 1/20 0.42
NSD2 O96028 1/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
ALDH1A1 P00352 2/20 0.42
TTR P02766 1/20 0.41
TDP1 Q9NUW8 2/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
ELANE P08246 1/20 0.40
TP53 P04637 1/20 0.40
CYP3A4 P08684 1/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1038715 0.91 BCL2 (0.80) BCL2MCL1MAOAMAOBADORA2A
SCHEMBL9925983 0.89 BCL2 (0.77) BCL2MCL1MAOAMAOBADORA2A
SCHEMBL7905103 0.85 BCL2 (0.70) BCL2MCL1MAOAMAOBMAPT
SCHEMBL12957364 0.83 BCL2 (0.69) BCL2MCL1MAOAMAOBADORA2A
SCHEMBL9239364 0.80 BCL2 (0.47) BCL2MCL1MAPTMAPK1MEN1
SCHEMBL8653360 0.79 BCL2 (0.73) BCL2MCL1MAOAMAOBMAPT
SCHEMBL12956976 0.79 BCL2 (0.76) BCL2MCL1MAOAMAOBMAPT
SCHEMBL9846537 0.78 ADORA2A (0.65) BCL2MCL1MAOAMAOBADORA2A
SCHEMBL9846493 0.78 ADORA2A (0.65) BCL2MCL1MAOAMAOBADORA2A
SCHEMBL9320566 0.77 MAOA (0.61) BCL2MCL1MAOAMAOBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0344110-B1 SUBSTITUTED NAPHTHACENES-5,12-DIONES AND THEIR USE CIBA-GEIGY AG (CH) 1992-09-16 EP disclosed
US-5001243-A Substituted naphthacene-5, 12-diones CIBA-GEIGY CORPORATION (US) 1991-03-19 US disclosed
EP-0344110-A2 Substituted naphthacenes-5,12-diones and their use CIBA-GEIGY AG (CH) 1989-11-29 EP disclosed