SCHEMBL9739172

SCHEMBL9739172

CN(C)c1nc(N)c2ncn(Cc3c(F)cccc3F)c2n1

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.51
ADORA1 P30542 1/20 0.51
PDE8A O60658 2/20 0.47
AXL P30530 2/20 0.45
MERTK Q12866 2/20 0.45
FLT3 P36888 1/20 0.45
TYRO3 Q06418 1/20 0.44
PDE4A P27815 2/20 0.44
PDE4B Q07343 2/20 0.44
PDE4C Q08493 2/20 0.44
PDE4D Q08499 2/20 0.44
CDK1 P06493 1/20 0.41
CCNB1 P14635 1/20 0.41
CCNE1 P24864 1/20 0.41
CDK2 P24941 1/20 0.41
PRKCA P17252 1/20 0.39
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3964946 0.87 ADORA2A (0.39) ADORA2AADORA1PDE8APDE4APDE4B
SCHEMBL9741263 0.87 ADORA2A (0.52) ADORA2AADORA1PDE8APDE4APDE4B
SCHEMBL9738800 0.86 PDE4A (0.50) ADORA2AADORA1AXLMERTKFLT3
SCHEMBL9740123 0.83 AXL (0.61) ADORA2AADORA1AXLMERTKFLT3
SCHEMBL9738975 0.83 ADORA2A (0.65) ADORA2AADORA1PDE8AAXLMERTK
SCHEMBL3959823 0.81 PDE8A (0.67) ADORA2AADORA1PDE8APDE4APDE4B
SCHEMBL7204383 0.81 PDE4A (0.62) ADORA2AADORA1PDE4APDE4BPDE4C
SCHEMBL9740849 0.81 ADORA2A (0.59) ADORA2AADORA1AXLMERTKFLT3
SCHEMBL9738479 0.81 AXL (0.53) ADORA2AADORA1PDE8AAXLMERTK
SCHEMBL9738741 0.79 ADORA2A (0.53) ADORA2AADORA1PDE8AAXLMERTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5110818-A Antiepileptic agents CIBA-GEIGY CORPORATION (US) 1992-05-05 US disclosed
EP-0363320-A2 Substituted 9H purine CIBA-GEIGY AG (CH) 1990-04-11 EP disclosed