SCHEMBL9739402

SCHEMBL9739402

O=C(O)c1[nH]c2cc(Cl)cc(Cl)c2c1CCN1CCN(c2ccccc2)C1=O

nearest known ligand 0.81

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 6/20 0.81
GPR17 Q13304 3/20 0.55
FBP1 P09467 1/20 0.55
HDAC1 Q13547 1/20 0.44
DRD2 P14416 2/20 0.43
DRD3 P35462 2/20 0.43
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9731518 0.94 GRIN1 (0.79) GRIN1GPR17FBP1HDAC1DRD2
SCHEMBL9732077 0.90 GRIN1 (1.00) GRIN1GPR17FBP1HDAC1
SCHEMBL9740502 0.90 GRIN1 (0.66) GRIN1GPR17FBP1HDAC1DRD2
SCHEMBL9732770 0.80 GRIN1 (0.69) GRIN1GPR17FBP1
SCHEMBL30559677 0.72 GPR17 (1.00) GRIN1GPR17FBP1
SCHEMBL8463078 0.72 GPR17 (1.00) GRIN1GPR17FBP1
SCHEMBL499308 0.71 GRIN1 (0.59) GRIN1GPR17
SCHEMBL499309 0.71 GRIN1 (0.59) GRIN1GPR17
SCHEMBL9731643 0.71 HDAC1 (0.45) GRIN1HDAC1DRD2DRD3KCNH2
SCHEMBL8603608 0.70 GRIN1 (0.56) GRIN1GPR17FBP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992020649-A2 SUBSTITUTED 2-CARBOXYINDOLES HAVING PHARMACEUTICAL ACTIVITY WARNER-LAMBERT COMPANY (US) 1992-11-26 WO claimed
WO-1992020649-A2 SUBSTITUTED 2-CARBOXYINDOLES HAVING PHARMACEUTICAL ACTIVITY WARNER-LAMBERT COMPANY (US) 1992-11-26 WO disclosed