SCHEMBL9740502

SCHEMBL9740502

COC(=O)c1[nH]c2cc(Cl)cc(Cl)c2c1CCN1CCN(c2ccccc2)C1=O

nearest known ligand 0.66

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 5/20 0.66
HDAC1 Q13547 2/20 0.43
FBP1 P09467 1/20 0.43
GPR17 Q13304 1/20 0.43
DRD2 P14416 7/20 0.40
DRD3 P35462 7/20 0.40
KCNH2 Q12809 6/20 0.40
DRD4 P21917 1/20 0.38
HTR2A P28223 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
MAPK1 P28482 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9739402 0.90 GRIN1 (0.81) GRIN1HDAC1FBP1GPR17DRD2
SCHEMBL9731518 0.84 GRIN1 (0.79) GRIN1HDAC1FBP1GPR17DRD2
SCHEMBL9732077 0.80 GRIN1 (1.00) GRIN1HDAC1FBP1GPR17MAPK1
SCHEMBL9732770 0.72 GRIN1 (0.69) GRIN1FBP1GPR17HPGDMAPK1
SCHEMBL9731682 0.71 GRIN1 (0.54) GRIN1FBP1GPR17
SCHEMBL9730824 0.71 GRIN1 (0.64) GRIN1FBP1GPR17KDM4EALDH1A1
SCHEMBL8416073 0.67 DRD2 (0.55) HDAC1DRD2DRD3KCNH2KDM4E
SCHEMBL9731504 0.67 GRIN1 (0.53) GRIN1FBP1GPR17MAPT
SCHEMBL9731643 0.66 HDAC1 (0.45) GRIN1HDAC1DRD2DRD3KCNH2
SCHEMBL499309 0.64 GRIN1 (0.59) GRIN1GPR17MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992020649-A2 SUBSTITUTED 2-CARBOXYINDOLES HAVING PHARMACEUTICAL ACTIVITY WARNER-LAMBERT COMPANY (US) 1992-11-26 WO claimed
WO-1992020649-A2 SUBSTITUTED 2-CARBOXYINDOLES HAVING PHARMACEUTICAL ACTIVITY WARNER-LAMBERT COMPANY (US) 1992-11-26 WO disclosed