SCHEMBL9739639

SCHEMBL9739639

Cc1c(Cc2ccccc2)oc2cc3c(cc12)OCO3

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 1/20 0.40
ALOX5 P09917 1/20 0.40
PTGS1 P23219 2/20 0.40
PTGS2 P35354 2/20 0.40
ALDH1A1 P00352 3/20 0.39
HPGD P15428 3/20 0.39
KDM4E B2RXH2 3/20 0.39
POLB P06746 1/20 0.39
TSHR P16473 3/20 0.39
LMNA P02545 1/20 0.39
MAPK1 P28482 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
GAA P10253 2/20 0.39
GLA P06280 1/20 0.39
HSD17B3 P37058 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ERAP1 Q9NZ08 1/20 0.39
MAOB P27338 2/20 0.38
GPR55 Q9Y2T6 3/20 0.38
CNR2 P34972 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9739636 0.79 KDM4E (0.36) ALOX5ALDH1A1HPGDKDM4EPOLB
SCHEMBL9739837 0.78 MAOB (0.48) ALOX5ALDH1A1HPGDKDM4EPOLB
SCHEMBL2546876 0.75 NQO1 (0.43) ALOX5ALDH1A1HPGDKDM4EPOLB
SCHEMBL31683019 0.74 KDM4E (0.46) ALOX5ALDH1A1HPGDKDM4EPOLB
SCHEMBL31683270 0.72 KDM4E (0.48) ALOX5ALDH1A1HPGDKDM4ESMN1; SMN2
SCHEMBL31683133 0.71 KDM4E (0.47) ALDH1A1HPGDKDM4EPOLBSMN1; SMN2
SCHEMBL2547565 0.71 NQO1 (0.42) ALDH1A1HPGDKDM4EPOLBLMNA
SCHEMBL2551423 0.68 NQO1 (0.35) ALOX5ALDH1A1HPGDKDM4EPOLB
SCHEMBL31683226 0.67 KDM4E (0.49) ALDH1A1HPGDKDM4EPOLBLMNA
SCHEMBL1422874 0.66 ALDH1A1 (0.58) ALDH1A1HPGDMAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5087638-A Inhibitors of mammalian leukotriene biosynthesis MERCK FROSST CANADA, INC. (CA) 1992-02-11 US disclosed
EP-0338782-A1 Benzofuran derivatives MERCK FROSST CANADA INC. (CA) 1989-10-25 EP disclosed
US-4863958-A TREATING ALLERGIC CONDITIONS, ASTHMA, CARDIOVASCULAR DISORDERS, AND INFLAMMATION MERCK FROSST CANADA, INC. (CA) 1989-09-05 US disclosed
EP-0165810-B1 BENZOFURAN AND BENZOTHIOPHENE DERIVATIVES, THEIR USE IN INHIBITING MAMMALIAN LEUKOTRIENE BIOSYNTHESIS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE DERIVATIVES MERCK FROSST CANADA INC. (CA) 1989-08-23 EP disclosed
EP-0165810-A2 Benzofuran and benzothiophene derivatives, their use in inhibiting mammalian leukotriene biosynthesis, and pharmaceutical compositions containing these derivatives MERCK FROSST CANADA INC. (CA) 1985-12-27 EP disclosed