SCHEMBL9739636

SCHEMBL9739636

Cc1c(Cc2ccccc2)oc2cc3c(cc12)OOC3

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
POLB P06746 1/20 0.36
HPGD P15428 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
HSD17B3 P37058 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ERAP1 Q9NZ08 1/20 0.36
ALOX5 P09917 2/20 0.35
NQO1 P15559 1/20 0.34
GPR55 Q9Y2T6 2/20 0.33
PTPN1 P18031 1/20 0.33
ALDH1A2 O94788 1/20 0.32
ALDH1B1 P30837 1/20 0.32
ALDH1A3 P47895 1/20 0.32
MAOB P27338 4/20 0.32
MTNR1A P48039 2/20 0.32
MTNR1B P49286 2/20 0.32
MAP2K1 Q02750 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9739639 0.79 CCR4 (0.40) KDM4EALDH1A1POLBHPGDGLA
SCHEMBL9739837 0.74 MAOB (0.48) KDM4EALDH1A1POLBHPGDGLA
SCHEMBL2546876 0.71 NQO1 (0.43) KDM4EALDH1A1POLBHPGDGLA
SCHEMBL31683019 0.70 KDM4E (0.46) KDM4EALDH1A1POLBHPGDGLA
SCHEMBL31683270 0.69 KDM4E (0.48) KDM4EALDH1A1HPGDGLAGAA
SCHEMBL11695911 0.68 IDH1 (0.42) ALDH1A1
SCHEMBL31683133 0.68 KDM4E (0.47) KDM4EALDH1A1POLBHPGDGLA
SCHEMBL11541643 0.67 ALOX5 (0.30) ALOX5
SCHEMBL31683226 0.63 KDM4E (0.49) KDM4EALDH1A1POLBHPGDGLA
SCHEMBL11538061 0.63 PIN1 (0.44) KDM4EALDH1A1POLBHPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5087638-A Inhibitors of mammalian leukotriene biosynthesis MERCK FROSST CANADA, INC. (CA) 1992-02-11 US disclosed
EP-0338782-A1 Benzofuran derivatives MERCK FROSST CANADA INC. (CA) 1989-10-25 EP disclosed
US-4863958-A TREATING ALLERGIC CONDITIONS, ASTHMA, CARDIOVASCULAR DISORDERS, AND INFLAMMATION MERCK FROSST CANADA, INC. (CA) 1989-09-05 US disclosed
EP-0165810-B1 BENZOFURAN AND BENZOTHIOPHENE DERIVATIVES, THEIR USE IN INHIBITING MAMMALIAN LEUKOTRIENE BIOSYNTHESIS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE DERIVATIVES MERCK FROSST CANADA INC. (CA) 1989-08-23 EP disclosed
EP-0165810-A2 Benzofuran and benzothiophene derivatives, their use in inhibiting mammalian leukotriene biosynthesis, and pharmaceutical compositions containing these derivatives MERCK FROSST CANADA INC. (CA) 1985-12-27 EP disclosed