SCHEMBL9740238

SCHEMBL9740238

COc1ccc(CCCN2CCCCC2C(C)N2CCc3cc(OC)c(OC)cc3CC2=O)cc1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 0.42
HCN4 Q9Y3Q4 2/20 0.41
MAPT P10636 1/20 0.41
CYP3A4 P08684 1/20 0.41
ALOX15 P16050 1/20 0.41
GAA P10253 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HRH3 Q9Y5N1 2/20 0.38
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
ABCC1 P33527 1/20 0.37
ABCG2 Q9UNQ0 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4D Q08499 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9740197 0.99 CYP3A4 (0.42) ABCB1HCN4MAPTCYP3A4ALOX15
SCHEMBL9740418 0.95 ABCB1 (0.46) ABCB1HCN4MAPTCYP3A4ALOX15
Hydrochloric Acid SCHEMBL9740153 0.94 ABCB1 (0.45) ABCB1HCN4MAPTCYP3A4ALOX15
SCHEMBL9739500 0.92 HCN4 (0.41) ABCB1HCN4MAPTCYP3A4ALOX15
SCHEMBL9739319 0.88 SMN1; SMN2 (0.42) ABCB1HCN4MAPTCYP3A4ALOX15
SCHEMBL9739180 0.87 SMN1; SMN2 (0.43) ABCB1HCN4MAPTCYP3A4ALOX15
Hydrochloric Acid SCHEMBL9739564 0.87 CYP3A4 (0.41) ABCB1HCN4MAPTCYP3A4ALOX15
SCHEMBL9739355 0.87 SMN1; SMN2 (0.42) GAASMN1; SMN2
SCHEMBL9740219 0.87 HCN4 (0.49) HCN4MAPTCYP3A4ALOX15GAA
SCHEMBL9740167 0.86 MTNR1B (0.43) GAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0224794-B1 CYCLIC AMINE DERIVATIVES, MEDICINES CONTAINING THESE COMPOUNDS AND PROCESS FOR THEIR PREPARATION Dr. Karl Thomae GmbH (DE) 1990-09-12 EP disclosed
EP-0224794-A2 Cyclic amine derivatives, medicines containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1987-06-10 EP disclosed