SCHEMBL9740282

SCHEMBL9740282

[c]1ccc2c(c1-c1ccncc1)OCO2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIPK3 Q9Y572 2/20 0.37
ROCK1 Q13464 2/20 0.33
PRKACA P17612 1/20 0.33
MAPT P10636 2/20 0.32
LMNA P02545 2/20 0.32
GAA P10253 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
PABPC1 P11940 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
HSD17B10 Q99714 1/20 0.32
FYN P06241 1/20 0.31
CASP3 P42574 1/20 0.31
SENP7 Q9BQF6 1/20 0.31
AHR P35869 1/20 0.31
DYRK1A Q13627 1/20 0.30
ROCK2 O75116 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL161183 0.82 ABCG2 (0.39) ALDH1A1HSD17B10CYP3A4
SCHEMBL8638641 0.80 MAPT (0.39) MAPTLMNAGAAKDM4EALDH1A1
SCHEMBL9738660 0.77 KDM4E (0.41) ROCK1PRKACAMAPTLMNAKDM4E
SCHEMBL6784931 0.75 HSP90AA1 (0.30)
SCHEMBL6210971 0.70 PDE4A (0.41) MAPTLMNAALDH1A1CYP3A4CYP2D6
SCHEMBL4347210 0.69 RIPK3 (0.56) RIPK3ROCK1MAPTALDH1A1DYRK1A
SCHEMBL3404505 0.69 ABCG2 (0.37) ALDH1A1HSD17B10CYP3A4
SCHEMBL83574 0.67 NQO2 (0.40) LMNAGAAALDH1A1CYP3A4CYP2D6
SCHEMBL6904035 0.67 ABCG2 (0.36) ALDH1A1HSD17B10
SCHEMBL6216565 0.66 ITGB2 (0.39) MAPTLMNAGAAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5134150-A Administering diaryl-substituted imidazothiazoles; antiarthritic agents SMITHKLINE BEECHAM CORPORATION (US) 1992-07-28 US disclosed