SCHEMBL9740511

SCHEMBL9740511

COc1cccc(CCN2CCC(CN3CCc4cc(OC)c(OC)cc4CC3=O)C2)c1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DHCR7 Q9UBM7 1/20 0.51
HTR1A P08908 2/20 0.48
SLC6A4 P31645 2/20 0.48
SIGMAR1 Q99720 1/20 0.47
MAPT P10636 1/20 0.47
HCN4 Q9Y3Q4 1/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
CYP3A4 P08684 1/20 0.46
ALOX15 P16050 1/20 0.46
HRH3 Q9Y5N1 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9740763 0.95 MEN1 (0.53) DHCR7SIGMAR1MAPTHCN4MEN1
Hydrochloric Acid SCHEMBL9740787 0.94 MEN1 (0.52) DHCR7SIGMAR1MAPTHCN4MEN1
SCHEMBL10720589 0.91 BCHE (0.47) DHCR7HTR1ASLC6A4MAPTHCN4
SCHEMBL9739547 0.90 ABCB1 (0.53) HTR1ASLC6A4MAPTHCN4CYP3A4
SCHEMBL9739280 0.89 HCN4 (0.59) DHCR7HTR1ASLC6A4MAPTHCN4
SCHEMBL9739687 0.86 HCN4 (0.45) DHCR7HTR1ASLC6A4MAPTHCN4
SCHEMBL9740561 0.85 CHRNB2 (0.49) SIGMAR1MAPTHCN4MEN1KMT2A
Hydrochloric Acid SCHEMBL9739300 0.85 CYP3A4 (0.46) MAPTHCN4MEN1KMT2ACYP3A4
SCHEMBL9746442 0.85 CHRNB2 (0.46) SIGMAR1MAPTHCN4CYP3A4ALOX15
SCHEMBL9739498 0.85 ABCB1 (0.51) MAPTHCN4MEN1KMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0224794-B1 CYCLIC AMINE DERIVATIVES, MEDICINES CONTAINING THESE COMPOUNDS AND PROCESS FOR THEIR PREPARATION Dr. Karl Thomae GmbH (DE) 1990-09-12 EP disclosed
EP-0224794-A2 Cyclic amine derivatives, medicines containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1987-06-10 EP disclosed