SCHEMBL9740561

SCHEMBL9740561

COc1cc2c(cc1OC)CC(=O)N(CC1CCCN(CCc3ccccc3)C1)CC2

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.49
CHRNB4 P30926 1/20 0.49
CHRNA3 P32297 1/20 0.49
CHRNA4 P43681 1/20 0.49
MAPT P10636 1/20 0.46
HCN4 Q9Y3Q4 1/20 0.46
CYP3A4 P08684 1/20 0.45
ALOX15 P16050 1/20 0.45
GAA P10253 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ABCB1 P08183 1/20 0.42
ABCG2 Q9UNQ0 1/20 0.42
CCR2 P41597 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
SIGMAR1 Q99720 1/20 0.41
LTA4H P09960 1/20 0.41
EPHX2 P34913 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9739064 0.99 CHRNB2 (0.48) CHRNB2CHRNB4CHRNA3CHRNA4MAPT
SCHEMBL9746442 0.97 CHRNB2 (0.46) CHRNB2CHRNB4CHRNA3CHRNA4MAPT
SCHEMBL9739855 0.95 CHRNB2 (0.46) CHRNB2CHRNB4CHRNA3CHRNA4MAPT
SCHEMBL9739720 0.94 CCR2 (0.47) CHRNB2CHRNB4CHRNA3CHRNA4MAPT
SCHEMBL9740796 0.94 CHRNB2 (0.45) CHRNB2CHRNB4CHRNA3CHRNA4MAPT
SCHEMBL9739409 0.94 CHRNB2 (0.47) CHRNB2CHRNB4CHRNA3CHRNA4MAPT
SCHEMBL9739498 0.92 ABCB1 (0.51) MAPTHCN4CYP3A4ALOX15GAA
SCHEMBL9741202 0.92 HCN4 (0.47) CHRNB2CHRNB4CHRNA3CHRNA4MAPT
SCHEMBL9739687 0.91 HCN4 (0.45) CHRNB2CHRNB4CHRNA3CHRNA4MAPT
SCHEMBL9740763 0.91 MEN1 (0.53) MAPTHCN4CYP3A4ALOX15MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0224794-A2 Cyclic amine derivatives, medicines containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1987-06-10 EP disclosed