SCHEMBL9745451

SCHEMBL9745451

COc1ccc2cc(C#Cc3ccc(C)cc3)ccc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.50
APP P05067 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2A6 P11509 1/20 0.48
RELA Q04206 1/20 0.46
AR P10275 1/20 0.45
NQO1 P15559 1/20 0.45
GRM5 P41594 2/20 0.44
CA12 O43570 2/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA9 Q16790 2/20 0.43
HSD17B1 P14061 1/20 0.43
HSD17B2 P37059 1/20 0.43
KCNH2 Q12809 1/20 0.42
HPGDS O60760 1/20 0.41
MAOB P27338 1/20 0.41
RAD52 P43351 1/20 0.41
CA7 P43166 1/20 0.41
CA14 Q9ULX7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9742128 0.95 HSD17B1 (0.47) ACHEAPPCYP1A2CYP2A6RELA
SCHEMBL9743076 0.90 APP (0.59) APPCYP1A2CYP2A6NQO1GRM5
SCHEMBL9742321 0.85 APP (0.53) APPCYP1A2CYP2A6NQO1CA12
SCHEMBL17086882 0.85 CYP1A2 (0.59) APPCYP1A2CYP2A6NQO1GRM5
SCHEMBL10525794 0.84 ACHE (0.71) ACHEAPPRELAARGRM5
SCHEMBL26828160 0.82 APP (0.64) ACHEAPPRELAARGRM5
SCHEMBL9744218 0.82 ESR1 (0.50) APPCYP1A2CYP2A6NQO1HPGDS
SCHEMBL17086858 0.82 CYP1A2 (0.60) APPCYP1A2CYP2A6NQO1GRM5
SCHEMBL13335288 0.81 CA12 (0.62) ACHEGRM5CA12CA1CA2
SCHEMBL11470578 0.81 CYP1A2 (0.52) APPCYP1A2CYP2A6NQO1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5084204-A Naphthylacetylenes MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-01-28 US disclosed