SCHEMBL9745831

SCHEMBL9745831

COCCOCOc1c(Br)cc(C=O)cc1OC

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.59
MAPK1 P28482 1/20 0.59
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
HTT P42858 2/20 0.46
HPGD P15428 2/20 0.46
MAPT P10636 5/20 0.43
LMNA P02545 2/20 0.43
FDPS P14324 1/20 0.42
SMN1; SMN2 Q16637 4/20 0.40
RAB9A P51151 2/20 0.40
NPC1 O15118 1/20 0.40
TNFRSF1A P19438 3/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TUBB1 Q9H4B7 3/20 0.39
TUBB4A P04350 1/20 0.39
TUBB P07437 1/20 0.39
TUBA3C P0DPH7 1/20 0.39
TUBA1B P68363 1/20 0.39
TUBA4A P68366 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7960002 0.93 ALDH1A1 (0.50) ALDH1A1MAPK1MEN1KMT2AHTT
SCHEMBL2709918 0.90 FDPS (0.47) ALDH1A1MAPK1MEN1KMT2AHTT
SCHEMBL6943688 0.89 ALDH1A1 (0.64) ALDH1A1MAPK1MEN1KMT2AHTT
SCHEMBL7962228 0.87 FDPS (0.45) ALDH1A1MAPK1MEN1KMT2AHTT
SCHEMBL31359168 0.87 ALDH1A1 (0.66) ALDH1A1MAPK1MEN1KMT2AHTT
SCHEMBL7437188 0.85 TNFRSF1A (0.47) ALDH1A1MAPK1MEN1KMT2AHTT
SCHEMBL7951806 0.83 FDPS (0.41) ALDH1A1MAPK1MEN1KMT2AHTT
SCHEMBL2649949 0.80 ALDH1A1 (0.64) ALDH1A1MAPK1MEN1KMT2AHTT
SCHEMBL9719099 0.80 ALDH1A1 (0.68) ALDH1A1MAPK1MEN1KMT2AHTT
SCHEMBL23202773 0.80 ALDH1A1 (0.56) ALDH1A1MAPK1MEN1KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0215250-B1 2-SUBSTITUTED-1,4-DIHYDROPYRIDINES, METHOD FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1992-12-30 EP disclosed
US-4845113-A USEFUL IN RADICAL SCAVENGING THERAPY BOEHRINGER BIOCHEMIA ROBIN S.P.A. (IT) 1989-07-04 US disclosed
EP-0215250-A1 2-Substituted-1,4-dihydropyridines, method for their preparation and pharmaceutical compositions containing them BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1987-03-25 EP disclosed