SCHEMBL9746606

SCHEMBL9746606

CC[C@H]1CC[C@H]2[C@@H]3[C@H](C)Cc4cc(OC(C)=O)ccc4[C@@]3(O)[C@@H](O)C[C@]12C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 4/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
LMNA P02545 2/20 0.40
ESR1 P03372 2/20 0.40
ADORA3 P0DMS8 2/20 0.40
ATM Q13315 2/20 0.40
PGR P06401 1/20 0.40
AR P10275 1/20 0.40
CHRM1 P11229 1/20 0.40
TBXA2R P21731 1/20 0.40
ADRA1A P35348 1/20 0.40
SLC6A3 Q01959 1/20 0.40
CYP3A4 P08684 2/20 0.35
MAPT P10636 2/20 0.35
TP53 P04637 1/20 0.35
NR1H2 P55055 2/20 0.34
NR1H3 Q13133 2/20 0.34
OPRD1 P41143 2/20 0.33
AKR1C3 P42330 1/20 0.33
OPRK1 P41145 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9746143 0.84 ESR1 (0.46) OPRM1SMN1; SMN2LMNAESR1ADORA3
SCHEMBL8775793 0.79 AKR1C3 (0.49) OPRM1SMN1; SMN2LMNAESR1ADORA3
SCHEMBL8775770 0.66 AKR1C3 (0.56) OPRM1SMN1; SMN2LMNAESR1ADORA3
SCHEMBL8775742 0.65 ESR1 (0.52) OPRM1SMN1; SMN2LMNAESR1ADORA3
SCHEMBL9747178 0.65 ESR1 (0.76) OPRM1SMN1; SMN2LMNAESR1ADORA3
SCHEMBL1688726 0.64 ESR1 (0.59) OPRM1SMN1; SMN2LMNAESR1ADORA3
SCHEMBL9746981 0.60 AKR1C3 (0.54) OPRM1SMN1; SMN2LMNAESR1ADORA3
SCHEMBL14827326 0.60 OPRM1 (0.55) OPRM1SMN1; SMN2LMNACYP3A4MAPT
SCHEMBL8775747 0.59 ESR1 (0.70) OPRM1SMN1; SMN2LMNAESR1ADORA3
SCHEMBL23765855 0.59 ESR1 (0.62) OPRM1SMN1; SMN2LMNAESR1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE34136-E Morning-after contraceptives SRI INTERNATIONAL (US) 1992-12-01 US disclosed
US-4859370-A 9 alpha, 11 beta-substituted and 11 beta-substituted estranes SRI INTERNATIONAL (US) 1989-08-22 US disclosed
US-4705783-A 9α, 11β-substituted and 11β-substituted estranes SRI INTERNATIONAL (US) 1987-11-10 US disclosed