SCHEMBL9747728

SCHEMBL9747728

Clc1ccc(Cn2cncn2)c(Cl)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.55
CCR2 P41597 1/20 0.55
CCR4 P51679 1/20 0.55
CYP3A4 P08684 2/20 0.54
CYP2C9 P11712 1/20 0.54
CYP19A1 P11511 6/20 0.50
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
LMNA P02545 1/20 0.46
PKM P14618 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP1A2 P05177 1/20 0.46
MAPT P10636 1/20 0.46
GABRA1 P14867 1/20 0.46
HPGD P15428 1/20 0.46
TSHR P16473 1/20 0.46
GABRG2 P18507 1/20 0.46
GABRB3 P28472 1/20 0.46
KDM4E B2RXH2 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14370854 0.84 KDM4E (0.50) CCR1CCR2CCR4CYP3A4CYP2C9
SCHEMBL7445529 0.84 CCR1 (0.50) CCR1CCR2CCR4CYP19A1MEN1
SCHEMBL9202589 0.84 BRD4 (0.51) CCR1CCR2CCR4CYP19A1MEN1
SCHEMBL8936736 0.81 CYP19A1 (0.53) CCR1CCR2CCR4CYP3A4CYP2C9
SCHEMBL3158915 0.81 CYP19A1 (0.50) CCR1CCR2CCR4CYP19A1KMT2A
SCHEMBL940881 0.79 CYP19A1 (0.62) CCR1CCR2CCR4CYP19A1MEN1
SCHEMBL2353053 0.78 KMT2A (0.49) CCR1CCR2CCR4CYP3A4CYP2C9
SCHEMBL10510964 0.78 MEN1 (0.55) CCR1CCR2CCR4CYP3A4CYP2C9
SCHEMBL7450404 0.78 CCR1 (0.51) CCR1CCR2CCR4CYP19A1MEN1
SCHEMBL10809801 0.78 LMNA (0.54) CCR1CCR2CCR4CYP3A4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5100890-A Antidepressants, Fungicides HOECHST AKTIENGESELLSCHAFT (DE) 1992-03-31 US disclosed
EP-0218118-B1 ARYLMETHYL AZOLES AND THEIR SALTS, METHOD FOR THEIR PREPARATION, COMPOSITIONS CONTAINING THEM AND THEIR USE HOECHST AKTIENGESELLSCHAFT (DE) 1991-09-18 EP disclosed
US-5023357-A Arylmethylazole preparation processes HOECHST AKTIENGESELLSCHAFT (DE) 1991-06-11 US disclosed
US-4876354-A FUNGICIDES, ANTIDEPRESSANTS HOECHST AKTIENGESELLSCHAFT (DE) 1989-10-24 US disclosed
EP-0218118-A1 Arylmethyl azoles and their salts, method for their preparation, compositions containing them and their use HOECHST AKTIENGESELLSCHAFT (DE) 1987-04-15 EP disclosed