SCHEMBL9748925

SCHEMBL9748925

CCCCOc1c(NCCCO)c(=O)c1=O

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADAMTS5 Q9UNA0 2/20 0.39
MAPT P10636 3/20 0.36
ALDH1A1 P00352 2/20 0.36
GAA P10253 2/20 0.35
THRA P10827 1/20 0.34
THRB P10828 1/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
ACHE P22303 6/20 0.33
POLB P06746 1/20 0.33
RAD52 P43351 1/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ITGB1 P05556 1/20 0.33
ITGA4 P13612 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9749261 0.84 ADAMTS5 (0.36) ADAMTS5MAPTALDH1A1GAATHRA
SCHEMBL9749443 0.81 NPC1 (0.35) ADAMTS5MAPTALDH1A1GAAPOLB
SCHEMBL31225285 0.79 GAA (0.42) MAPTALDH1A1GAAPOLBNPC1
SCHEMBL8592976 0.78 MAPT (0.43) MAPTALDH1A1GAAPOLBMEN1
SCHEMBL25025146 0.76 POLB (0.41) MAPTALDH1A1GAAPOLB
SCHEMBL22301648 0.76 POLB (0.41) MAPTALDH1A1GAAPOLB
SCHEMBL31163657 0.76 POLB (0.41) MAPTALDH1A1GAAPOLB
SCHEMBL22895170 0.75 GAA (0.46) MAPTALDH1A1GAATHRBPOLB
SCHEMBL9749005 0.74 ALDH1A1 (0.43) ADAMTS5MAPTALDH1A1
SCHEMBL7887050 0.74 SMN1; SMN2 (0.41) ADAMTS5MAPTALDH1A1GAATHRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0294615-B1 CYCLOBUTENE-3,4-DIONE-INTERMEDIATES AND THEIR USE IN THE PREPARATION OF HISTAMINE H2-ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 1992-04-15 EP disclosed
US-4927970-A Substituted 3-cyclobutene-1,2-dione intermediates BRISTOL-MYERS COMPANY (US) 1990-05-22 US disclosed
EP-0294615-A1 Cyclobutene-3,4-dione-intermediates and their use in the preparation of histamine h2-antagonists Bristol-Myers Squibb Company (US) 1988-12-14 EP disclosed