SCHEMBL9749313

SCHEMBL9749313

C=CCOc1ccccc1OC(C)=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LIG1 P18858 1/20 0.54
HSD17B10 Q99714 3/20 0.49
HPGD P15428 2/20 0.49
TSHR P16473 2/20 0.49
MAPK1 P28482 1/20 0.49
ADRB2 P07550 2/20 0.48
ADRB1 P08588 2/20 0.48
LMNA P02545 2/20 0.48
CYP1A2 P05177 2/20 0.48
SLC22A1 O15245 1/20 0.48
HTR1A P08908 1/20 0.48
CYP2D6 P10635 1/20 0.48
HTR2A P28223 1/20 0.48
SLC6A4 P31645 1/20 0.48
ADRA1A P35348 1/20 0.48
PTGS1 P23219 2/20 0.48
PTGS2 P35354 8/20 0.47
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 1/20 0.47
ESR1 P03372 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7924944 0.87 LIG1 (0.51) LIG1HSD17B10HPGDTSHRMAPK1
SCHEMBL29168887 0.86 LIG1 (0.57) LIG1HSD17B10HPGDTSHRMAPK1
SCHEMBL29168888 0.84 LIG1 (0.55) LIG1HSD17B10HPGDTSHRMAPK1
SCHEMBL6686762 0.83 KDM4E (0.47) LIG1TSHRMAPK1ADRB2ADRB1
SCHEMBL8754763 0.82 ALDH1A1 (0.54) LIG1HSD17B10HPGDTSHRMAPK1
1-Allyloxy-2-Methoxybenzene SCHEMBL27937762 0.81 POLB (0.57) LIG1HSD17B10HPGDTSHRMAPK1
1,2-Diallyloxybenzene SCHEMBL366516 0.81 HPGD (0.60) LIG1HSD17B10HPGDTSHRMAPK1
1,2-Diallyloxybenzene SCHEMBL29768784 0.81 HPGD (0.60) LIG1HSD17B10HPGDTSHRMAPK1
SCHEMBL10451271 0.81 LIG1 (0.46) LIG1HSD17B10HPGDTSHRMAPK1
SCHEMBL2032188 0.80 PTGS2 (0.52) HSD17B10HPGDTSHRMAPK1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105555759-A Compounds with antibacterial activity FUND MEDINA CT DE EXCELENCIA EN INVESTIG DE MEDICAMENTOS INNOVADORES EN ANDALUCIA 2016-05-04 CN disclosed
CN-101903367-B Antitumor compounds PHARMA MAR, S.A. (ES) 2015-08-05 CN disclosed
CN-102190643-B Antitumoral compounds PHARMA MAR SA 2015-02-25 CN disclosed
CN-101932592-B Antitumoral compounds PHARMA MAR SA 2014-02-26 CN disclosed
CN-103038240-A Synthetic method for preparing ecteinascidin compounds PHARMA MAR SA 2013-04-10 CN disclosed
CN-102190643-A Antitumoral compounds PHARMA MAR SA 2011-09-21 CN disclosed
CN-101932592-A Antineoplastic compound PHARMA MAR SA 2010-12-29 CN disclosed
CN-101903367-A Antitumor compounds PHARMA MAR SA 2010-12-01 CN disclosed
EP-0230475-B1 NOVEL UREA DERIVATIVES, PROCESSES FOR PRODUCTION THEREOF AND HERBICIDE MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1992-03-18 EP disclosed
EP-0169581-B1 ANTITUSSIVE AND MUCUS REGULATING 2-SUBSTITUTED THIAZOLIDINES BOEHRINGER BIOCHEMIA ROBIN S.p.A. (IT) 1989-12-06 EP disclosed
US-4857643-A Antitussive and mucus regulating 2-substituted thiazolidines BOEHRINGER BIOCHEMIA ROBIN S.P.A. (IT) 1989-08-15 US disclosed
US-4838924-A NONPHYTOTOXIC MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1989-06-13 US disclosed
US-4798898-A BRONCHODILATORS BOEHRINGER BIOCHEMIA ROBIN S.P.A. (IT) 1989-01-17 US disclosed
EP-0169581-A2 Antitussive and mucus regulating 2-substituted thiazolidines BOEHRINGER BIOCHEMIA ROBIN S.p.A. (IT) 1986-01-29 EP disclosed
US-4310527-A DISORDERS OF CAROIAC RHYTHM AND CORONARY HEART DISEASES AND HYDPERTENSION CIBA-GEIGY CORPORATION (US) 1982-01-12 US disclosed
US-4140789-A ADRENERGIC BLOCKING AGENTS, CARDIOTONIC, ANTIARRHYTHMIA, HYPOTENSIVE CIBA-GEIGY CORPORATION (US) 1979-02-20 US disclosed