SCHEMBL9749813

SCHEMBL9749813

CCC(Cc1nsnc1OCC(O)CN(O)C(C)(C)C)C(=O)O

nearest known ligand 0.32

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.32
BLM P54132 1/20 0.32
CYP1A2 P05177 1/20 0.30
ADRB2 P07550 1/20 0.30
ADRB1 P08588 1/20 0.30
CYP3A4 P08684 1/20 0.30
HTR1A P08908 1/20 0.30
CYP2D6 P10635 1/20 0.30
ADRB3 P13945 1/20 0.30
NFKB1 P19838 1/20 0.30
DRD1 P21728 1/20 0.30
SIGMAR1 Q99720 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9749858 0.81 SMN1; SMN2 (0.49) SMN1; SMN2BLMCYP1A2ADRB2ADRB1
SCHEMBL9749331 0.78 ADRB2 (0.40) BLMCYP1A2ADRB2ADRB1CYP3A4
SCHEMBL11033838 0.69 ADRB2 (0.49) SMN1; SMN2BLMCYP1A2ADRB2ADRB1
SCHEMBL11753852 0.61 CYP2D6 (0.57) SMN1; SMN2BLMCYP1A2ADRB2ADRB1
SCHEMBL11756802 0.59 CYP2D6 (0.46) SMN1; SMN2BLMCYP1A2ADRB2ADRB1
SCHEMBL11755467 0.57 ADRB2 (0.46) ADRB2ADRB1CYP2D6ADRB3
SCHEMBL11403374 0.56 CYP2D6 (0.59) SMN1; SMN2BLMCYP1A2ADRB2ADRB1
SCHEMBL25846983 0.55 CA2 (0.48) TDP1
Chloromethane SCHEMBL28143162 0.55 CA2 (0.64) TDP1
SCHEMBL6114 0.55

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0131006-B1 ESTERS OF 3-(3-SUBSTITUTED-AMINO-2-HYDROXYPROPOXY)-4-SUBSTITUTED-1,2,5-THIADIAZOLE DERIVATIVES THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1992-06-10 EP claimed