SCHEMBL9750113

SCHEMBL9750113

C=C1N(C)c2ccc(Oc3cccc(OC)c3)cc2C1(C)C

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRIA2 P42262 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.44
POLB P06746 3/20 0.42
MTNR1B P49286 4/20 0.38
MTNR1A P48039 3/20 0.38
MAPT P10636 1/20 0.38
BACE1 P56817 2/20 0.37
AADAT Q8N5Z0 1/20 0.37
KDM4E B2RXH2 1/20 0.36
PGR P06401 3/20 0.36
MPI P34949 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9750257 0.90 GRIA2 (0.42) GRIA2SMN1; SMN2POLBMAPTMPI
SCHEMBL3819871 0.90 MAPT (0.43) POLBMAPTKDM4EMPITDP1
SCHEMBL8942200 0.87 GRIA2 (0.42) GRIA2BACE1MPITDP1
SCHEMBL9750440 0.82 GRIA2 (0.42) GRIA2SMN1; SMN2POLBMAPTKDM4E
SCHEMBL9750442 0.81 TDP1 (0.37) SMN1; SMN2POLBMAPTBACE1MPI
Questiomycin B SCHEMBL9330595 0.79 ALDH1A1 (0.41) SMN1; SMN2POLBMAPTBACE1KDM4E
SCHEMBL4602650 0.78 TDP1 (0.41) MAPTKDM4EMPITDP1
SCHEMBL5851872 0.75 MEN1 (0.37) SMN1; SMN2POLBMAPTBACE1KDM4E
SCHEMBL5850476 0.75 CYP1A1 (0.48) MAPTBACE1TDP1
SCHEMBL22245096 0.75 SMN1; SMN2 (0.56) GRIA2SMN1; SMN2POLBMTNR1BMTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5120858-A Condensation of 2-methyleneindoline and formic acid in acetic anhydride MILES INC. (US) 1992-06-09 US disclosed
EP-0058863-B1 PROCESS FOR THE PREPARATION OF TRIMETHINE DYESTUFFS BAYER AG (DE) 1985-01-23 EP disclosed
US-4419511-A Process for the preparation of trimethine dyestuffs BAYER AKTIENGESELLSCHAFT (US) 1983-12-06 US disclosed
EP-0058863-A1 Process for the preparation of trimethine dyestuffs BAYER AG (DE) 1982-09-01 EP disclosed