SCHEMBL9750374

SCHEMBL9750374

O=C(O)c1cn(C2CC2)c2c3c(c(F)cc2c1=O)N1CCC[C@H]1CO3

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AADAT Q8N5Z0 2/20 0.58
KDM4E B2RXH2 5/20 0.57
ALDH1A1 P00352 4/20 0.57
HPGD P15428 3/20 0.57
HSD17B10 Q99714 3/20 0.57
ALB P02768 1/20 0.57
HRH3 Q9Y5N1 1/20 0.57
POLB P06746 3/20 0.56
TUBB4A P04350 1/20 0.56
TUBB P07437 1/20 0.56
TUBA3C P0DPH7 1/20 0.56
TUBA1B P68363 1/20 0.56
TUBA4A P68366 1/20 0.56
TUBB4B P68371 1/20 0.56
TUBB3 Q13509 1/20 0.56
TUBB2A Q13885 1/20 0.56
TUBB8 Q3ZCM7 1/20 0.56
TUBA3E Q6PEY2 1/20 0.56
TUBA1A Q71U36 1/20 0.56
SLC47A1 Q96FL8 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL116382 1.00 AADAT (0.58) AADATKDM4EALDH1A1HPGDHSD17B10
SCHEMBL115248 0.91 AADAT (0.53) AADATKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9750378 0.88 AADAT (0.45) AADATKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9749840 0.86 AADAT (0.51) AADATKDM4EALDH1A1HPGDHSD17B10
SCHEMBL10424507 0.86 KDM4E (0.55) AADATKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9749826 0.86 KDM4E (0.52) AADATKDM4EALDH1A1HPGDHSD17B10
SCHEMBL12825263 0.86 AADAT (0.54) AADATKDM4EALDH1A1HPGDHSD17B10
SCHEMBL116181 0.85 ALDH1A1 (0.52) AADATKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9749825 0.84 AADAT (0.48) AADATKDM4EALDH1A1HPGDHSD17B10
SCHEMBL584176 0.84 AADAT (0.52) AADATKDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0216345-B1 QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1992-02-19 EP disclosed
US-4977265-A WITH BACTERICIDAL ACTIVITY HOFFMANN-LA ROCHE INC. (US) 1990-12-11 US disclosed
US-4946847-A BACTERICIDES HOFFMANN-LA ROCHE INC. (US) 1990-08-07 US disclosed
US-4806541-A ANTIBACTERIAL AGENTS HOFFMANN-LA ROCHE INC. (US) 1989-02-21 US disclosed
EP-0216345-A2 Quinoline derivatives F. HOFFMANN-LA ROCHE AG (CH) 1987-04-01 EP disclosed