SCHEMBL9751699

SCHEMBL9751699

Fc1ccc(C2C[CH]CCC2)cc1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HTR2B P41595 1/20 0.37
USP30 Q70CQ3 1/20 0.35
KDM1A O60341 2/20 0.35
MAOB P27338 1/20 0.35
GRIA4 P48058 1/20 0.35
SLC6A2 P23975 2/20 0.33
SLC6A4 P31645 2/20 0.33
SLC6A3 Q01959 2/20 0.33
CYP2D6 P10635 1/20 0.33
KCNH2 Q12809 1/20 0.33
HCAR2 Q8TDS4 1/20 0.32
USP5 P45974 2/20 0.32
HDAC6 Q9UBN7 1/20 0.32
CHRNB2 P17787 1/20 0.31
ADRA2C P18825 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
CHRNA7 P36544 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9185425 0.81 HTR2A (0.41) HTR2AHTR2CHTR2BUSP30KDM1A
SCHEMBL12917832 0.81 GRIA4 (0.43) HTR2AHTR2CHTR2BUSP30KDM1A
SCHEMBL27887265 0.79 ATM (0.38) HTR2AHTR2CHTR2BKDM1ASLC6A2
SCHEMBL127034 0.79 ACMSD (0.44) HTR2AHTR2CHTR2BACMSD
SCHEMBL29389392 0.76 HTR2A (0.46) HTR2AHTR2CHTR2BUSP30KDM1A
SCHEMBL808710 0.76 HTR2A (0.46) HTR2AHTR2CHTR2BUSP30KDM1A
SCHEMBL27417610 0.76 HTR3A (0.48) SLC6A2SLC6A3
SCHEMBL9184228 0.75 HTR2A (0.37) HTR2AHTR2CHTR2BUSP30KDM1A
SCHEMBL17186857 0.75 SLC6A2 (0.39) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL9184233 0.75 HTR2A (0.37) HTR2AHTR2CHTR2BUSP30KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438574-A1 2,5-DISUBSTITUTED HETEROCYCLES AND MESOMORPHOUS MEDIUM. MERCK PATENT GMBH (DE) 1991-07-31 EP disclosed
EP-0438575-A1 BENZOL DERIVATIVES AND LIQUID CRYSTALLINE MEDIUM. MERCK PATENT GMBH (DE) 1991-07-31 EP disclosed
WO-1991002710-A2 BENZOL DERIVATIVES AND LIQUID CRYSTALLINE MEDIUM MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1991-03-07 WO disclosed
WO-1991002780-A1 2,5-DISUBSTITUTED HETEROCYCLES AND MESOMORPHOUS MEDIUM MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1991-03-07 WO disclosed