SCHEMBL9752026

SCHEMBL9752026

O=C(C=Cc1ccc(Br)cc1)ON1C(=O)CCC1=O

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.42
ESR2 Q92731 1/20 0.42
GPR183 P32249 9/20 0.42
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
MAPT P10636 2/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.40
SLC5A1 P13866 1/20 0.40
SLC5A2 P31639 1/20 0.40
KCNH2 Q12809 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP1B1 Q16678 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9390893 0.86 CA12 (0.54) ESR1ESR2MAOBRAB9A
SCHEMBL14546443 0.86 CA12 (0.54) ESR1ESR2MAOBRAB9A
SCHEMBL9411957 0.85 CYP1A2 (0.50) MAOAMAOBMAPTALDH1A1CYP1A2
SCHEMBL9411954 0.85 CYP1A2 (0.50) MAOAMAOBMAPTALDH1A1CYP1A2
SCHEMBL9551400 0.85 HSD11B1 (0.50) GPR183MAOAMAOBMAPTALDH1A1
SCHEMBL9551421 0.85 MAPT (0.47) MAOAMAOBMAPTALDH1A1CYP1A2
SCHEMBL1711201 0.84 LMNA (0.47) MAOAMAOBMAPTALDH1A1CYP1A2
SCHEMBL7882197 0.84 LMNA (0.47) MAOAMAOBMAPTALDH1A1CYP1A2
SCHEMBL10381850 0.82 F3 (0.55) GPR183MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL13967398 0.81 KDM4E (0.53) MAPTALDH1A1NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0449884-A4 DERIVATIVES OF TETRAPEPTIDES AS CCK AGONISTS 1991-10-30 EP disclosed
EP-0449884-A1 DERIVATIVES OF TETRAPEPTIDES AS CCK AGONISTS ABBOTT LABORATORIES (US) 1991-10-09 EP disclosed
WO-1990006937-A1 DERIVATIVES OF TETRAPEPTIDES AS CCK AGONISTS ABBOTT LABORATORIES (US) 1990-06-28 WO disclosed