SCHEMBL9752144

SCHEMBL9752144

CC(=O)Nc1ccc2c(c1)CC(N)CC2

nearest known ligand 0.60

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.54
DRD3 P35462 2/20 0.54
ACHE P22303 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9776821 0.81 MTNR1A (0.51) ACHE
SCHEMBL10447740 0.80 DRD2 (0.58) DRD2DRD3ACHE
Hydrochloric Acid SCHEMBL10447759 0.79 DRD2 (0.57) DRD2DRD3ACHE
SCHEMBL9776895 0.78 DRD3 (0.50) DRD2DRD3ACHE
SCHEMBL2463176 0.78 MTNR1A (0.60) ACHE
SCHEMBL9776892 0.77 DRD2 (0.49) DRD2DRD3
SCHEMBL2246315 0.76 CYP1A2 (0.54)
SCHEMBL9776896 0.76 DRD2 (0.64) DRD2DRD3
SCHEMBL2245582 0.76 BAZ2B (0.64)
SCHEMBL1673429 0.76 BAZ2B (0.69)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5053430-A For treating schizophrenia BOEHRINGER INGELHEIM KG (DE) 1991-10-01 US disclosed
EP-0435988-A1 2-AMINO-7-CARBAMOYL-1,2,3,4-TETRAHYDRONAPHTHALENES, PROCESS FOR PREPARING THEM AND THEIR USE AS DRUGS BOEHRINGER INGELHEIM KG (DE) 1991-07-10 EP disclosed
WO-1991001297-A1 2-AMINO-7-CARBAMOYL-1,2,3,4-TETRAHYDRONAPHTHALENES, PROCESS FOR PREPARING THEM AND THEIR USE AS DRUGS BOEHRINGER INGELHEIM KG (DE) 1991-02-07 WO disclosed
EP-0361300-A1 Use of 2,7 diamino-1,2,3,4-tetrahydronaphthalenes as drugs, 2,7 diamino-1,2,3,4-tetrahydronaphthalenes as well as processes for their preparation BOEHRINGER INGELHEIM KG (DE) 1990-04-04 EP disclosed