SCHEMBL9752647

SCHEMBL9752647

CC(CCCCN)N(C)S(=O)(=O)c1cccc2c(N(C)C)cccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.54
CYP2C19 P33261 1/20 0.54
HTT P42858 1/20 0.54
HIF1A Q16665 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
CA2 P00918 1/20 0.52
F2 P00734 3/20 0.46
PRSS1 P07477 3/20 0.46
PRSS2 P07478 3/20 0.46
PRSS3 P35030 3/20 0.46
EDNRA P25101 5/20 0.44
KMT2A Q03164 1/20 0.43
ATM Q13315 1/20 0.43
HTR7 P34969 3/20 0.42
DAPK3 O43293 1/20 0.40
DYRK3 O43781 1/20 0.40
ROCK2 O75116 1/20 0.40
RPS6KA5 O75582 1/20 0.40
PRKD3 O94806 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4270202 0.80 CA2 (0.52) CYP1A2CYP2C19HTTHIF1ATDP1
SCHEMBL5508602 0.80 CYP1A2 (0.64) CYP1A2CYP2C19HTTHIF1ATDP1
SCHEMBL9455666 0.77 CYP1A2 (0.57) CYP1A2CYP2C19HTTHIF1ATDP1
SCHEMBL6416698 0.76 CA2 (0.57) CYP1A2CYP2C19HTTHIF1ATDP1
SCHEMBL30597369 0.76 CYP1A2 (0.45) CYP1A2CYP2C19HTTHIF1ATDP1
SCHEMBL19270962 0.76 CYP1A2 (0.71) CYP1A2CYP2C19HTTHIF1ATDP1
SCHEMBL9779598 0.75 EDNRA (0.48) CA2F2PRSS1PRSS2PRSS3
SCHEMBL6254983 0.75 CYP1A2 (0.41) CYP1A2CYP2C19HTTHIF1ATDP1
SCHEMBL597354 0.75 MMP2 (0.54) F2
SCHEMBL319321 0.75 MMP2 (0.54) F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991010427-A2 THE EFFECT OF TRANSGLUTAMINASE INHIBITION ON MICROFILARIAE DEVELOPMENT AND MACROFILARIAE VIABILITY BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1991-07-25 WO disclosed
WO-1989001512-A1 A SPONGE ENZYME HAVING TRANSGLUTAMINASE-LIKE ACTIVITY THE LIPOSOME COMPANY, INC. (US) 1989-02-23 WO disclosed