SCHEMBL9753622

SCHEMBL9753622

O=C(O)c1cn2c(C(=O)O)cccc2n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 3/20 0.53
PTGS2 P35354 3/20 0.53
KDM4E B2RXH2 6/20 0.45
ALOX15 P16050 1/20 0.45
TSHR P16473 1/20 0.45
ACMSD Q8TDX5 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
GAA P10253 1/20 0.44
GNE Q9Y223 1/20 0.40
GLA P06280 1/20 0.38
ATM Q13315 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38
TGFBR1 P36897 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8608104 0.85 PTGS1 (0.46) PTGS1PTGS2KDM4EALOX15TSHR
SCHEMBL4542221 0.84 GAA (0.48) PTGS1PTGS2KDM4EALOX15TSHR
SCHEMBL4536170 0.81 GAA (0.48) PTGS1PTGS2KDM4EGAAGLA
SCHEMBL3035988 0.81 PTGS1 (0.51) PTGS1PTGS2KDM4EALOX15TSHR
SCHEMBL119204 0.81 PTGS1 (0.51) PTGS1PTGS2KDM4EALOX15TSHR
SCHEMBL21816403 0.81 TGFBR1 (0.44) PTGS1PTGS2KDM4EGAAGLA
SCHEMBL3306389 0.81 PTGS1 (0.51) PTGS1PTGS2KDM4EALOX15TSHR
SCHEMBL119926 0.81 GAA (0.66) PTGS1PTGS2KDM4EALOX15TSHR
SCHEMBL8606782 0.78 PTGS1 (0.49) PTGS1PTGS2KDM4EALOX15TSHR
SCHEMBL7872399 0.78 MAP2K1 (0.51) PTGS1PTGS2KDM4ETSHRTGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0436831-A2 Imidazo[1,2-a]pyridinylalkyl compounds for treatment of neurotoxic injury G.D. Searle & Co. (US) 1991-07-17 EP claimed
WO-1991008211-A1 IMIDAZO[1,2-a]PYRIDINYLALKYL COMPOUNDS FOR TREATMENT OF NEUROTOXIC INJURY G.D. SEARLE & CO. (US) 1991-06-13 WO claimed
EP-0436831-A2 Imidazo[1,2-a]pyridinylalkyl compounds for treatment of neurotoxic injury G.D. Searle & Co. (US) 1991-07-17 EP disclosed
WO-1991008211-A1 IMIDAZO[1,2-a]PYRIDINYLALKYL COMPOUNDS FOR TREATMENT OF NEUROTOXIC INJURY G.D. SEARLE & CO. (US) 1991-06-13 WO disclosed